SCHEMBL7205577

SCHEMBL7205577

COCCOc1cc2ncnc(C3C(=O)Nc4ccc(F)cc43)c2cc1OC

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 17/20 0.46
EGFR P00533 1/20 0.43
FGFR1 P11362 1/20 0.43
FLT1 P17948 1/20 0.43
FLT4 P35916 1/20 0.43
TRPA1 O75762 1/20 0.43
RET P07949 1/20 0.42
KIF5B P33176 1/20 0.42
MAPK7 Q13164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7210197 0.89 FBP1 (0.51) KDRFGFR1FLT1
SCHEMBL7205793 0.88 KDR (0.48) KDRFGFR1FLT1
Hydrochloric Acid SCHEMBL7209976 0.88 KDR (0.47) KDREGFR
SCHEMBL7211312 0.86 KDR (0.42) KDREGFRFGFR1FLT1MAPK7
SCHEMBL7207079 0.86 KDR (0.44) KDREGFR
SCHEMBL4518666 0.86 PDGFRB (0.46) KDREGFRFGFR1FLT1FLT4
Hydrochloric Acid SCHEMBL7212863 0.86 KDR (0.42) KDREGFRFGFR1FLT1MAPK7
Hydrochloric Acid SCHEMBL7210078 0.86 KDR (0.43) KDREGFR
SCHEMBL7211368 0.86 ABCG2 (0.43) KDRFGFR1FLT1
Hydrochloric Acid SCHEMBL7206364 0.86 CHEK1 (0.46) KDREGFRFGFR1FLT1FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912557-B1 OXINDOLE DERIVATIVES ASTRAZENECA AB (SE) 2003-07-09 EP claimed
US-6265411-B1 ANGIOGENESIS INHIBITOR ZENECA LIMITED (GB) 2001-07-24 US claimed
EP-0912557-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1999-05-06 EP claimed
WO-1997042187-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1997-11-13 WO claimed
EP-0912557-B1 OXINDOLE DERIVATIVES ASTRAZENECA AB (SE) 2003-07-09 EP disclosed
US-6265411-B1 ANGIOGENESIS INHIBITOR ZENECA LIMITED (GB) 2001-07-24 US disclosed
EP-0912557-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1999-05-06 EP disclosed
WO-1997042187-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1997-11-13 WO disclosed