SCHEMBL7207232

SCHEMBL7207232

CCc1ccnc(C(=O)c2[nH]c3ccc(C(F)(F)F)cc3c2CC(=O)OC)c1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.65
PTGS1 P23219 7/20 0.55
EGFR P00533 2/20 0.43
CDK2 P24941 1/20 0.40
BCHE P06276 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
AKR1C3 P42330 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6169961 0.90 PTGS2 (0.76) PTGS2PTGS1EGFRCDK2MEN1
SCHEMBL27554774 0.89 PTGS2 (0.68) PTGS2PTGS1EGFR
SCHEMBL27554775 0.89 PTGS2 (0.67) PTGS2PTGS1EGFRCDK2BCHE
SCHEMBL27533987 0.88 PTGS2 (0.83) PTGS2PTGS1MEN1KMT2A
SCHEMBL27533827 0.86 PTGS2 (0.60) PTGS2PTGS1MEN1KMT2A
SCHEMBL27554906 0.83 PTGS2 (0.80) PTGS2PTGS1EGFRCDK2
SCHEMBL8113137 0.82 PTGS2 (0.55) PTGS2PTGS1EGFRCDK2BCHE
SCHEMBL27532185 0.81 PTGS2 (0.61) PTGS2PTGS1AKR1C3
SCHEMBL27554509 0.80 PTGS2 (0.58) PTGS2PTGS1
SCHEMBL6168900 0.79 PTGS2 (1.00) PTGS2PTGS1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1284064-A 2,3-substituted indole compounds as cox-2 inhibitors PFIZER PHARMA (US) 2001-02-14 CN claimed
US-6608070-B1 Useful for treatment of medical condition in which prostaglandins are implicated as pathogens NAKAO KAZUNARI (JP) 2003-08-19 US disclosed
CN-1284064-A 2,3-substituted indole compounds as cox-2 inhibitors PFIZER PHARMA (US) 2001-02-14 CN disclosed