SCHEMBL7208047

SCHEMBL7208047

Cc1cccc2c(Br)cc(O)nc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
TP53 P04637 2/20 0.42
HTT P42858 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
USP2 O75604 1/20 0.42
HSP90AA1 P07900 1/20 0.42
PDE7A Q13946 1/20 0.42
PARP1 P09874 2/20 0.41
ELANE P08246 1/20 0.41
RAD52 P43351 3/20 0.41
GAA P10253 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
TNKS O95271 2/20 0.40
TNKS2 Q9H2K2 2/20 0.40
PARP2 Q9UGN5 1/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29631413 0.83 KDM4E (0.51) KDM4EMEN1KMT2ATP53HTT
SCHEMBL935117 0.83 KDM4E (0.51) KDM4EMEN1KMT2ATP53HTT
SCHEMBL7219924 0.81 TP53 (0.54) KDM4EMEN1KMT2ATP53HTT
SCHEMBL7218856 0.81 ELANE (0.43) KDM4EMEN1KMT2ATP53HTT
SCHEMBL11401006 0.81 PARP1 (0.43) KDM4EMEN1KMT2ATP53HTT
SCHEMBL30612099 0.79 MAPT (0.47) KDM4EMEN1KMT2ATP53HTT
SCHEMBL26103062 0.79 MAPT (0.47) KDM4EMEN1KMT2ATP53HTT
SCHEMBL7208150 0.76 MAPT (0.54) KDM4EMEN1KMT2ATP53HTT
SCHEMBL6806506 0.75 ELANE (0.47) KDM4EMEN1KMT2ATP53HTT
SCHEMBL9849276 0.75 TNKS (0.47) KDM4EMEN1KMT2ATP53HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6608085-B1 Administering for neuroprotection VERNALIS RESEARCH LIMITED (GB) 2003-08-19 US disclosed
EP-1107761-A2 4-QUINOLINEMETHANOL DERIVATIVES AS PURINE RECEPTOR ANTAGONISTS (II) VERNALIS RESEARCH LIMITED (GB) 2001-06-20 EP disclosed
WO-2000013682-A2 4-QUINOLINEMETHANOL DERIVATIVES AS PURINE RECEPTOR ANTAGONISTS.(II) VERNALIS RESEARCH LIMITED (GB) 2000-03-16 WO disclosed