SCHEMBL7208436

SCHEMBL7208436

Cc1ccc(Sc2nc(N)c3nc(Br)n(Cc4ccccc4)c3n2)cc1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.55
ADORA1 P30542 5/20 0.55
TMIGD3 P0DMS9 3/20 0.46
ADORA2B P29275 3/20 0.46
TSHR P16473 2/20 0.43
ALDH1A1 P00352 2/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
TLR7 Q9NYK1 10/20 0.41
NPSR1 Q6W5P4 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7211495 0.92 ADORA2A (0.61) ADORA2AADORA1TMIGD3ADORA2BTSHR
SCHEMBL7209443 0.86 TSHR (0.45) ADORA2AADORA1TSHRALDH1A1POLB
SCHEMBL7205651 0.86 ADORA2A (0.55) ADORA2AADORA1TMIGD3ADORA2BTSHR
SCHEMBL7210266 0.84 ADORA2A (0.61) ADORA2AADORA1TMIGD3ADORA2BTSHR
SCHEMBL7204591 0.82 ADORA2A (0.58) ADORA2AADORA1TMIGD3ADORA2BTSHR
SCHEMBL7211539 0.81 ADORA2A (0.57) ADORA2AADORA1TMIGD3ADORA2BTSHR
SCHEMBL7205103 0.81 ADORA2A (0.60) ADORA2AADORA1TMIGD3ADORA2BTSHR
SCHEMBL7210598 0.81 ADORA2A (0.54) ADORA2AADORA1TMIGD3ADORA2BTSHR
SCHEMBL7205682 0.81 ADORA2A (0.56) ADORA2AADORA1TMIGD3ADORA2BTLR7
SCHEMBL5732024 0.80 ADORA2A (0.65) ADORA2AADORA1TMIGD3ADORA2BTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1035123-B1 NOVEL HETEROCYCLIC COMPOUNDS SUMITOMO PHARMA (JP) 2003-08-20 EP disclosed
US-6329381-B1 INTERFERONS, VIRICIDES AND ANTICARCINOGENIC AGENTS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1035123-A1 NOVEL HETEROCYCLIC COMPOUNDS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-09-13 EP disclosed