SCHEMBL7208712

SCHEMBL7208712

CCC(CO)Nc1nc(Nc2cccc(OC)c2)c2ncn(CC)c2n1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 10/20 0.73
CDK5 Q00535 11/20 0.60
CDK5R1 Q15078 10/20 0.60
KDM4E B2RXH2 1/20 0.60
NPC1 O15118 1/20 0.60
POLB P06746 1/20 0.60
MAPT P10636 1/20 0.60
CCNA2 P20248 10/20 0.55
CDK2 P24941 10/20 0.55
CSNK1A1 P48729 2/20 0.55
CCNT1 O60563 1/20 0.55
CCNB1 P14635 1/20 0.55
CCNE1 P24864 1/20 0.55
CDK7 P50613 1/20 0.55
CDK9 P50750 1/20 0.55
CCNH P51946 1/20 0.55
MNAT1 P51948 1/20 0.55
GSK3B P49841 1/20 0.55
CCNA1 P78396 9/20 0.54
DYRK1A Q13627 8/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5840807 1.00 CDK1 (0.73) CDK1CDK5CDK5R1KDM4ENPC1
SCHEMBL5841668 0.87 CDK5 (0.78) CDK1CDK5CDK5R1KDM4ENPC1
SCHEMBL8710243 0.87 CDK5 (0.78) CDK1CDK5CDK5R1KDM4ENPC1
SCHEMBL5841752 0.87 CDK1 (0.72) CDK1CDK5CDK5R1KDM4ENPC1
SCHEMBL5841742 0.87 CDK1 (0.72) CDK1CDK5CDK5R1KDM4ENPC1
SCHEMBL8706894 0.87 CDK5 (0.78) CDK1CDK5CDK5R1KDM4ENPC1
SCHEMBL5839851 0.85 CDK1 (0.67) CDK1CDK5CDK5R1KDM4ENPC1
SCHEMBL5839860 0.85 CDK1 (0.67) CDK1CDK5CDK5R1KDM4ENPC1
SCHEMBL5839334 0.85 CDK1 (0.68) CDK1CDK5CDK5R1KDM4ENPC1
SCHEMBL5839344 0.85 CDK1 (0.68) CDK1CDK5CDK5R1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874846-B1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 2003-04-02 EP disclosed