SCHEMBL7208988

SCHEMBL7208988

CC(C)(C)OOC(=O)O.NCCCN

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 2/20 0.36
CYP1A2 P05177 2/20 0.36
THRB P10828 2/20 0.36
BLM P54132 2/20 0.36
KMT2A Q03164 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
GABRR3 A8MPY1 1/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
HDAC3 O15379 1/20 0.36
GABBR2 O75899 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRR1 P24046 1/20 0.36
GABRB3 P28472 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrazine SCHEMBL28251779 0.84 TSHR (0.45) TSHRALDH1A1HSD17B10TDP1
SCHEMBL209234 0.83
SCHEMBL3861871 0.71 PAOX (0.48) TDP1KMT2AMEN1PAOX
SCHEMBL27344240 0.70 TSHR (0.38) TSHRALDH1A1HSD17B10TDP1LMNA
SCHEMBL1899004 0.69 TSHR (0.40) TSHRALDH1A1HSD17B10TDP1
Propane SCHEMBL2296352 0.68 TSHR (0.36) TSHRALDH1A1HSD17B10TDP1
SCHEMBL11121471 0.68 TSHR (0.41) TSHRALDH1A1HSD17B10TDP1
Butylamine SCHEMBL3926203 0.68 DNM1 (0.37) TSHRALDH1A1LMNACYP1A2THRB
SCHEMBL22733774 0.67 TSHR (0.39) TSHRALDH1A1HSD17B10TDP1
Acetic Acid SCHEMBL4397846 0.67 CYP1A2 (0.53) TSHRALDH1A1LMNACYP1A2THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000072-B1 PROCESS FOR THE PREPARATION OF [2-((8,9)- DIOXO-2,6-DIAZABICYCLO [5.2.0]-NON-1(7)-EN-2-YL)-ETHYL] PHOSPHONIC ACID WYETH CORP (US) 2003-02-19 EP disclosed
EP-1000072-A1 PROCESS FOR THE PREPARATION OF 2-((8,9)- DIOXO-2,6-DIAZABICYCLO 5.2.0]-NON-1(7)-EN-2-YL)-ETHYL] PHOSPHONIC ACID AMERICAN HOME PRODUCTS CORPORATION (US) 2000-05-17 EP disclosed
US-6011168-A Process for the preparation[2-((8,9)-dioxo-2,6-diazabicyclo[5.2.0]-non-1(7)-en-2-yl)ethy l]phosphonic acid AMERICAN HOME PRODUCTS CORPORATION (US) 2000-01-04 US disclosed
US-5990307-A Process for the preparation of [2-((8.9)-Dioxo-2,6-Diazabicyclo [5.2.0]-Non-1(7)-en-2yl) Ethyl]Phosphonic acid AMERICAN HOME PRODUCTS CORPORATION (US) 1999-11-23 US disclosed
WO-1999006417-A1 PROCESS FOR THE PREPARATION OF [2-((8,9)- DIOXO-2,6-DIAZABICYCLO [5.2.0]-NON-1(7)-EN-2-YL)-ETHYL] PHOSPHONIC ACID AMERICAN HOME PRODUCTS CORPORATION (US) 1999-02-11 WO disclosed