SCHEMBL7209159

SCHEMBL7209159

CC1(C)CC(NS(=O)(=O)c2ccc(OCc3ccc(F)cc3Cl)cc2)(C(=O)NO)CO1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 5/20 0.63
ADAMTS7 Q9UKP4 3/20 0.63
MMP13 P45452 12/20 0.57
MMP2 P08253 3/20 0.57
MMP14 P50281 3/20 0.57
ADAMTS4 O75173 2/20 0.57
MMP1 P03956 13/20 0.53
ADAM17 P78536 5/20 0.50
MMP3 P08254 2/20 0.50
MMP9 P14780 2/20 0.50
MMP8 P22894 2/20 0.50
TNF P01375 1/20 0.50
ADAMTS1 Q9UHI8 1/20 0.50
MMP12 P39900 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7208134 0.92 ADAMTS5 (0.62) ADAMTS5ADAMTS7MMP13MMP2MMP14
SCHEMBL7214318 0.91 ADAMTS5 (0.64) ADAMTS5ADAMTS7MMP13MMP2MMP14
SCHEMBL7208067 0.88 ADAMTS5 (0.61) ADAMTS5ADAMTS7MMP13MMP2MMP14
SCHEMBL7208610 0.88 ADAMTS5 (0.63) ADAMTS5ADAMTS7MMP13MMP2MMP14
SCHEMBL7208123 0.87 ADAMTS5 (0.58) ADAMTS5ADAMTS7MMP13MMP2MMP14
SCHEMBL7214222 0.86 ADAMTS5 (0.65) ADAMTS5ADAMTS7MMP13MMP2MMP14
SCHEMBL7214327 0.83 ADAMTS5 (0.59) ADAMTS5ADAMTS7MMP13MMP2MMP14
SCHEMBL7212992 0.83 ADAMTS5 (0.61) ADAMTS5ADAMTS7MMP13MMP2MMP14
SCHEMBL7213000 0.82 ADAMTS5 (0.66) ADAMTS5ADAMTS7MMP13MMP2MMP14
SCHEMBL7207007 0.81 ADAMTS5 (0.60) ADAMTS5ADAMTS7MMP13MMP2MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181285-B1 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PROD INC (US) 2003-10-08 EP disclosed
EP-1181285-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES Pfizer Products Inc. (US) 2002-02-27 EP disclosed
US-6342521-B1 DRUGS FOR TREATMENT OF ARTHRITIS PFIZER INC. 2002-01-29 US disclosed
WO-2000073294-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PRODUCTS INC. (US) 2000-12-07 WO disclosed