SCHEMBL7209338

SCHEMBL7209338

COc1cc(C2=NCCc3ccccc32)ccc1NS(=O)(=O)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA7 P43166 2/20 0.45
CA9 Q16790 2/20 0.45
CA14 Q9ULX7 2/20 0.45
STAT3 P40763 2/20 0.42
MAPK10 P53779 1/20 0.41
CCR9 P51686 3/20 0.41
PPIB P23284 1/20 0.41
PPIA P62937 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6718878 0.89 CCR9 (0.47) CA1CA2CA7CA9CA14
SCHEMBL6717992 0.87 STAT3 (0.42) STAT3CCR9CYP3A4CYP2D6PSEN1
SCHEMBL6716456 0.87 CA2 (0.47) CA1CA2CA7CA9CA14
SCHEMBL6716880 0.85 MEN1 (0.55) CA1CA2CA7CA9CA14
SCHEMBL6715116 0.84 CYP3A4 (0.49) CA1CA2CA7CA9CA14
SCHEMBL6716509 0.83 TP53 (0.49) CA1CA2CA7CA9CA14
SCHEMBL6717804 0.83 DDB1 (0.45) CA1CA2CA7CA9CA14
SCHEMBL6718026 0.77 CA1 (0.42) CA1CA2CA7CA9CA14
SCHEMBL6714720 0.77 MAPK10 (0.54) CA1CA2CA7CA9CA14
SCHEMBL6718234 0.77 CCR9 (0.51) CA1CA2CA7CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337515-A1 (DIHYDRO)ISOQUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 2003-08-27 EP disclosed
WO-2002040450-A1 (DIHYDRO)ISOQUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS ALTANA PHARMA AG (DE) 2002-05-23 WO disclosed