SCHEMBL7213533

SCHEMBL7213533

Oc1ccc(OC(Cc2ccccc2)C[C@]2(O)CCNC[C@H]2O)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
CDK7 P50613 1/20 0.35
CCNH P51946 1/20 0.35
MNAT1 P51948 1/20 0.35
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
ADRA1D P25100 2/20 0.35
ADRA1A P35348 2/20 0.35
ADRA1B P35368 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
PTGS1 P23219 1/20 0.33
SLC6A2 P23975 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7209171 1.00 CDK1 (0.35) CDK1CCNE1CDK2CDK7CCNH
SCHEMBL7214886 0.92 PPARG (0.43) LMNACYP1A2PTGS1SLC6A2CYP2C19
SCHEMBL7209167 0.92 PPARG (0.43) LMNACYP1A2PTGS1SLC6A2CYP2C19
SCHEMBL8195162 0.75 MAOB (0.44) LMNACYP1A2PTGS1SLC6A2CYP2C19
SCHEMBL8195227 0.75 MAOB (0.44) LMNACYP1A2PTGS1SLC6A2CYP2C19
SCHEMBL8487882 0.74 GRIN2D (0.37) GRIN2DGRIN3BADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL8482025 0.73 GRIN2D (0.36) GRIN2DGRIN3BADRA1DADRA1AADRA1B
SCHEMBL6376835 0.73 CDK7 (0.41) CDK1CCNE1CDK2CDK7CCNH
SCHEMBL7208859 0.73 CDK7 (0.41) CDK1CCNE1CDK2CDK7CCNH
SCHEMBL6382124 0.73 CDK7 (0.41) CDK1CCNE1CDK2CDK7CCNH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1278730-A2 4-BENZYL-1- 2-(4-HYDROXY-PHENOXY)-ETHYL]-PIPERIDINE-3,4-DIOL F. HOFFMANN-LA ROCHE AG (CH) 2003-01-29 EP claimed
WO-2001081309-A2 4-BENZYL-1-[2-(4-HYDROXY-PHENOXY)-ETHYL]-PIPERIDINE-3,4-DIOL F. HOFFMANN-LA ROCHE AG (CH) 2001-11-01 WO claimed
EP-1278730-A2 4-BENZYL-1- 2-(4-HYDROXY-PHENOXY)-ETHYL]-PIPERIDINE-3,4-DIOL F. HOFFMANN-LA ROCHE AG (CH) 2003-01-29 EP disclosed
WO-2001081309-A2 4-BENZYL-1-[2-(4-HYDROXY-PHENOXY)-ETHYL]-PIPERIDINE-3,4-DIOL F. HOFFMANN-LA ROCHE AG (CH) 2001-11-01 WO disclosed