SCHEMBL8487882

SCHEMBL8487882

Oc1ccc(OC(Cc2ccccc2)CC(O)C2(O)CCNCC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 2/20 0.37
GRIN3B O60391 2/20 0.37
ADRA1D P25100 2/20 0.37
ADRA1A P35348 2/20 0.37
ADRA1B P35368 2/20 0.37
GRIN1 Q05586 2/20 0.37
GRIN2A Q12879 2/20 0.37
GRIN2B Q13224 2/20 0.37
GRIN2C Q14957 2/20 0.37
GRIN3A Q8TCU5 2/20 0.37
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
PTGS1 P23219 1/20 0.35
SLC6A2 P23975 1/20 0.35
CYP2C19 P33261 1/20 0.35
PTGS2 P35354 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HIF1A Q16665 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
TACR1 P25103 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8482025 0.99 GRIN2D (0.36) GRIN2DGRIN3BADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL8485176 0.88 PPARG (0.33) GRIN2BSLC6A2PPARGPPARA
Hydrochloric Acid SCHEMBL8523937 0.80 ADRB2 (0.38) CYP1A2CYP2C19TSHR
Hydrochloric Acid SCHEMBL8487046 0.80 PRMT5 (0.37) CYP1A2CYP2C19
SCHEMBL8486004 0.80 ESR1 (0.39) GRIN2DGRIN3BADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL8486958 0.79 ESR1 (0.38) GRIN2DGRIN3BADRA1DADRA1AADRA1B
SCHEMBL7209171 0.74 CDK1 (0.35) GRIN2DGRIN3BADRA1DADRA1AADRA1B
SCHEMBL7213533 0.74 CDK1 (0.35) GRIN2DGRIN3BADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL10773246 0.69 LMNA (0.47) LMNACYP1A2PTGS1SLC6A2CYP2C19
SCHEMBL8482269 0.68 GRIN2D (0.41) GRIN2DGRIN3BADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889026-A 4-hydroxy-piperodine derivatives HOFFMANN-LA ROCHE INC. (US) 1999-03-30 US disclosed