SCHEMBL7216178

SCHEMBL7216178

CS(=O)(=O)c1ccc(-c2cccn2-c2ccc(O)cc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.74
PTGS1 P23219 3/20 0.55
ENPP2 Q13822 1/20 0.53
MELK Q14680 1/20 0.50
ALOX5 P09917 1/20 0.44
FYN P06241 1/20 0.43
MAP4K4 O95819 1/20 0.43
MINK1 Q8N4C8 1/20 0.43
TNIK Q9UKE5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7210560 1.00 PTGS2 (0.74) PTGS2PTGS1ENPP2MELKALOX5
SCHEMBL5311655 0.87 PTGS2 (0.76) PTGS2PTGS1ALOX5
SCHEMBL5312538 0.87 PTGS2 (0.76) PTGS2PTGS1ALOX5
SCHEMBL5312009 0.86 PTGS2 (0.76) PTGS2PTGS1ALOX5
SCHEMBL7211950 0.85 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL5309601 0.85 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL5309608 0.85 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL5314063 0.85 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL5310941 0.85 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL7210285 0.85 PTGS2 (0.74) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed
US-5935990-A PYRROLYL DERIVATIVES HAVING AT POSITION 1 OR 5 A PHENYL SUBSTITUTED WITH METHYLSULFONYL OR AMINOSULFONYL; INHIBIT CYCLOOXYGENASE-2 FOR USE TREATMENT OF INFLAMMATION, AS AN ANALGESIC, OR AS AN ANTIPYRETIC G.D. SEARLE & CO. (US) 1999-08-10 US disclosed