SCHEMBL7218266

SCHEMBL7218266

CNC(=O)ON=C(C)OC(=O)[C@@H](N)CCCCNOC(=O)NC

nearest known ligand 0.31

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 4/20 0.31
NOS1 P29475 3/20 0.31
NOS3 P29474 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
BLM P54132 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7225562 0.83 DPP7 (0.32)
SCHEMBL7909560 0.82 NOS2 (0.32) NOS2NOS1NOS3CYP1A2CYP3A4
SCHEMBL8821862 0.77 DPP7 (0.31)
SCHEMBL7908797 0.75 SMN1; SMN2 (0.36)
SCHEMBL7218187 0.72
SCHEMBL7218263 0.72 FOLH1 (0.38)
SCHEMBL7224578 0.70 DPP7 (0.33)
SCHEMBL7226863 0.69 NOS2 (0.46) NOS2NOS1NOS3CYP1A2CYP3A4
SCHEMBL7911329 0.69 NOS2 (0.46) NOS2NOS1NOS3CYP1A2CYP3A4
SCHEMBL7220182 0.68 DPP7 (0.32) NOS2NOS1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6576780-B1 Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors GD SEARLE & COMPANY 2003-06-10 US disclosed
US-6207708-B1 FOR THERAPY AND PROPHYLAXIS OF AUTOIMMUNE AND/OR INFLAMMATORY CONDITIONS AFFECTING THE JOINTS SUCH AS ARTHRITIS, AND INFLAMMATORY BOWEL DISEASE, CARDIVASCULAR ISCHEMIA, DIABETES, CONGESTIVE HEART FAILURE, MYOCARDITIS, ATHEROSCLEROSIS, G. D. SEARLE & COMPANY 2001-03-27 US disclosed
EP-0885188-B1 HYDROXYAMIDINO DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2000-09-27 EP disclosed