SCHEMBL7219741

SCHEMBL7219741

N#Cc1cncc(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.44
CYP11B2 P19099 3/20 0.44
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
KDR P35968 2/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
PLK4 O00444 1/20 0.43
CHEK1 O14757 1/20 0.43
AURKA O14965 1/20 0.43
CHUK O15111 1/20 0.43
ROCK2 O75116 1/20 0.43
CHEK2 O96017 1/20 0.43
INSR P06213 1/20 0.43
CDK1 P06493 1/20 0.43
CSF1R P07333 1/20 0.43
PIM1 P11309 1/20 0.43
FGFR1 P11362 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL169815 0.88 CYP11B1 (0.49) CYP11B1CYP11B2ADORA2AADORA1ALDH1A1
SCHEMBL3089783 0.81 ADORA2A (0.47) CYP11B1CYP11B2ADORA2AADORA1ALDH1A1
SCHEMBL5329333 0.80 ADORA2A (0.46) CYP11B1CYP11B2ADORA2AADORA1ALDH1A1
SCHEMBL5336784 0.77 PRKCQ (0.54) CYP11B1CYP11B2ADORA2AADORA1PRKCQ
SCHEMBL7220037 0.76 ADORA1 (0.49) ADORA2AADORA1ALDH1A1KDM4EHTT
SCHEMBL2978375 0.76 KDM5A (0.40) CYP11B1CYP11B2ADORA2AADORA1ALDH1A1
SCHEMBL1146097 0.76 CYP1A2 (0.57) CYP11B1CYP11B2ALDH1A1KDM4EHTT
SCHEMBL7215513 0.76 ATR (0.50) CYP11B1CYP11B2ALDH1A1KDM4EHTT
SCHEMBL565466 0.75 ESR2 (0.50) ALDH1A1KDM4EMAPTHTTNPSR1
SCHEMBL28598885 0.73 ATM (0.35) ADORA2AADORA1KDRMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603007-B1 Intermediates in the fields of pharmaceuticals, agrichemicals, ligands, silver halide photosensitive materials, liquid crystals, surfactants, electrophotography and organic electroluminescence SANKIO CHEMICAL CO., LTD. (JP) 2003-08-05 US disclosed
EP-1231207-A1 NOVEL BIPYRIDYL DERIVATIVES Sankio Chemical Co., Ltd. (JP) 2002-08-14 EP disclosed