SCHEMBL7220029

SCHEMBL7220029

CCCCc1cncc(C#N)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
RAF1 P04049 1/20 0.36
NPC1 O15118 2/20 0.35
HPGD P15428 2/20 0.35
RAB9A P51151 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CASP3 P42574 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21705943 0.93 TSHR (0.53) TSHRHSD17B10L3MBTL1TDP1HPGD
SCHEMBL26169758 0.93 TSHR (0.53) TSHRHSD17B10L3MBTL1TDP1HPGD
SCHEMBL7219748 0.89 PDCD1 (0.38) TSHRHSD17B10CHRNB2CHRNA4RAF1
SCHEMBL7213725 0.81 CYP2A6 (0.48) CHRNB2CHRNA4RAF1GRIN1GRIN2B
SCHEMBL10807925 0.80 TDP1 (0.50) TSHRCHRNB2CHRNA4L3MBTL1TDP1
SCHEMBL23783636 0.78 CHRNA7 (0.41) CHRNB2CHRNA4RAF1HTTGRIN1
SCHEMBL27209742 0.78 HRH3 (0.37) HSD17B10RAF1HPGDMAPK1GRIN1
SCHEMBL18728443 0.78 CYP11B1 (0.36) HSD17B10CHRNB2CHRNA4RAF1HPGD
SCHEMBL3508498 0.77 GRIN1 (0.35) CHRNB2CHRNA4RAF1GRIN1GRIN2B
SCHEMBL24615861 0.77 GRM5 (0.38) RAF1PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603007-B1 Intermediates in the fields of pharmaceuticals, agrichemicals, ligands, silver halide photosensitive materials, liquid crystals, surfactants, electrophotography and organic electroluminescence SANKIO CHEMICAL CO., LTD. (JP) 2003-08-05 US disclosed
EP-1231207-A1 NOVEL BIPYRIDYL DERIVATIVES Sankio Chemical Co., Ltd. (JP) 2002-08-14 EP disclosed
CN-1043760-C \"Pyridinecarboximidamide compounds and the use thereof\ KIRN BEER KABUSHIKI KAISHA (JP) 1999-06-23 CN disclosed
CN-1077949-A Pyridine carboxy imido acid amide compound and application thereof KIRIN BREWERY (JP) 1993-11-03 CN disclosed