SCHEMBL7219748

SCHEMBL7219748

CCCc1cncc(C#N)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 2/20 0.38
CD274 Q9NZQ7 2/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
RAF1 P04049 1/20 0.37
CYP2A6 P11509 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CYP19A1 P11511 1/20 0.36
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7220029 0.89 TSHR (0.44) PDCD1CD274CHRNB2CHRNA4RAF1
SCHEMBL21705943 0.86 TSHR (0.53) CYP19A1TSHRHSD17B10
SCHEMBL26169758 0.86 TSHR (0.53) CYP19A1TSHRHSD17B10
SCHEMBL7213725 0.84 CYP2A6 (0.48) PDCD1CD274CHRNB2CHRNA4RAF1
SCHEMBL23783636 0.81 CHRNA7 (0.41) CHRNB2CHRNA4RAF1CYP11B1CYP11B2
SCHEMBL18728443 0.81 CYP11B1 (0.36) CHRNB2CHRNA4RAF1CYP11B1CYP11B2
SCHEMBL27209742 0.81 HRH3 (0.37) RAF1CYP11B1CYP11B2HSD17B10
SCHEMBL24107273 0.80 GRIN1 (0.35) CHRNB2CHRNA4RAF1CYP11B1CYP11B2
SCHEMBL22778574 0.80 NOS1 (0.39) PDCD1CD274TSHRHSD17B10
SCHEMBL24615861 0.80 GRM5 (0.38) PDCD1CD274RAF1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4043461-A1 COMPOUND AS SMALL MOLECULE INHIBITOR PD-1/PD-L1 AND APPLICATION THEREOF Medshine Discovery Inc. (CN) 2022-08-17 EP disclosed
WO-2019046784-A1 COMPOUNDS AND METHODS FOR MODULATING ADENOSINE A2B RECEPTOR AND ADENOSINE A2A RECEPTOR CORVUS PHARMACEUTICALS, INC. (US) 2019-03-07 WO disclosed
US-6603007-B1 Intermediates in the fields of pharmaceuticals, agrichemicals, ligands, silver halide photosensitive materials, liquid crystals, surfactants, electrophotography and organic electroluminescence SANKIO CHEMICAL CO., LTD. (JP) 2003-08-05 US disclosed
EP-1231207-A1 NOVEL BIPYRIDYL DERIVATIVES Sankio Chemical Co., Ltd. (JP) 2002-08-14 EP disclosed