SCHEMBL7220958

SCHEMBL7220958

CCCn1c(=O)c2[nH]c(-c3ccc(OCC(=O)NCc4ccccc4)cc3)nc2n(CCC)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 12/20 1.00
ADORA2A P29274 11/20 1.00
ADORA3 P0DMS8 7/20 1.00
ADORA1 P30542 6/20 1.00
KDM4E B2RXH2 1/20 0.75
ALDH1A1 P00352 1/20 0.75
CYP3A4 P08684 1/20 0.75
MAPT P10636 1/20 0.75
HPGD P15428 1/20 0.75
ALOX15 P16050 1/20 0.75
PMP22 Q01453 1/20 0.75
SMN1; SMN2 Q16637 1/20 0.75
HSD17B10 Q99714 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7220779 0.88 ADORA2B (1.00) ADORA2BADORA2AADORA3ADORA1KDM4E
Xanthine Amine Congener SCHEMBL1000686 0.86 ADORA2A (1.00) ADORA2BADORA2AADORA3ADORA1KDM4E
SCHEMBL7227160 0.85 ADORA2B (1.00) ADORA2BADORA2AADORA3ADORA1KDM4E
SCHEMBL7235224 0.85 ADORA2B (1.00) ADORA2BADORA2AADORA3ADORA1
Xanthine Amine Congener SCHEMBL25227375 0.85 ADORA2A (0.98) ADORA2BADORA2AADORA3ADORA1KDM4E
Xanthine Amine Congener SCHEMBL15124872 0.85 ADORA2A (0.98) ADORA2BADORA2AADORA3ADORA1KDM4E
SCHEMBL7228029 0.84 ADORA2B (1.00) ADORA2BADORA2AADORA3ADORA1
SCHEMBL1065789 0.84 ADORA2B (0.73) ADORA2BADORA2AADORA3ADORA1KDM4E
SCHEMBL1223882 0.83 ADORA2B (1.00) ADORA2BADORA2AADORA3ADORA1KDM4E
SCHEMBL9159693 0.82 ADORA2A (0.77) ADORA2BADORA2AADORA3ADORA1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6545002-B1 Treating asthma, diarrhea, insulin resistance, diabetes, ischemia/reprefusion injuries, diabetic retinopathy or hyperbaric oxygen-induced retinopathy UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2003-04-08 US disclosed