SCHEMBL7222006

SCHEMBL7222006

Cn1cc2c(n1)-c1c(C(=O)Nc3ccc4c(n3)OCCO4)c[nH]c1CCC2

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.38
RAB9A P51151 6/20 0.38
PKM P14618 3/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
TYK2 P29597 2/20 0.33
DRD4 P21917 2/20 0.32
DRD2 P14416 1/20 0.32
HTR1F P30939 4/20 0.32
HTR1A P08908 2/20 0.31
WDR5 P61964 1/20 0.30
HTR1D P28221 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7216812 0.84 NPC1 (0.56) NPC1RAB9APKMALDH1A1LMNA
SCHEMBL7222852 0.79 NPC1 (0.43) NPC1RAB9APKMALDH1A1LMNA
SCHEMBL6834487 0.78 GAA (0.43) NPC1RAB9APKMALDH1A1DRD4
SCHEMBL7218324 0.78 MAPT (0.42) NPC1RAB9APKMALDH1A1LMNA
SCHEMBL7216813 0.77 F10 (0.39) NPC1RAB9A
SCHEMBL6834466 0.77 KMT2A (0.37) NPC1RAB9AALDH1A1DRD4DRD2
SCHEMBL7216265 0.76 NPC1 (0.38) NPC1RAB9AALDH1A1LMNA
SCHEMBL6834309 0.75 LMNA (0.42) NPC1RAB9APKMALDH1A1LMNA
SCHEMBL6831069 0.74 NAMPT (0.53) NPC1RAB9AALDH1A1
SCHEMBL6304803 0.74 DRD4 (0.44) ALDH1A1DRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6653471-B2 Tricyclic heteroaromatic compounds containing pyrrole ring; central nervous system disorder treatment; side effect reduction NEUROGEN CORPORATION 2003-11-25 US disclosed