SCHEMBL7222799

SCHEMBL7222799

C(=CC1CCc2ccccc21)c1ccon1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.34
PDPK1 O15530 1/20 0.34
CYP11B2 P19099 5/20 0.33
CYP19A1 P11511 4/20 0.33
CYP17A1 P05093 1/20 0.33
RECQL P46063 1/20 0.32
ADRA1A P35348 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
TAS1R2 Q8TE23 1/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11631174 0.70 PDPK1 (0.47) IDO1PDPK1CYP11B2ADRA1A
SCHEMBL11631168 0.70 PDPK1 (0.47) IDO1PDPK1CYP11B2ADRA1A
SCHEMBL28636065 0.70 IDO1 (0.43) IDO1PDPK1CYP11B2CA1CA2
SCHEMBL11882269 0.69 IDO1 (0.40) IDO1PDPK1CYP11B2CA1CA2
SCHEMBL9165650 0.66 IDO1 (0.46) IDO1PDPK1CYP11B2CYP19A1CYP17A1
SCHEMBL384149 0.66 IDO1 (0.46) IDO1PDPK1CYP11B2CYP19A1CYP17A1
SCHEMBL1567191 0.66 PDPK1 (0.50) IDO1PDPK1CYP11B2ADRA1A
SCHEMBL21937667 0.66 IDO1 (0.46) IDO1PDPK1CYP11B2CYP19A1CYP17A1
SCHEMBL22391437 0.66 IDO1 (0.50) IDO1PDPK1CYP11B2CYP19A1CYP17A1
SCHEMBL1567129 0.66 HTR1A (0.47) IDO1PDPK1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627652-B1 Treatment of diseases or conditions of the type which are normally treated with retinoid-like compounds is disclosed, with pharmaceutical compositions containing an active compound which is a selective agonist of the RXR retinoid ALLERGAN, INC. 2003-09-30 US disclosed
US-5475113-A Treatment of skin disorders, skin cancer ALLERGAN, INC. (US) 1995-12-12 US disclosed
EP-0682516-A1 THERAPEUTIC USE OF COMPOUNDS HAVING SELECTIVE AGONIST-LIKE ACTIVITY ON RXR RETINOID RECEPTORS ALLERGAN, INC. (US) 1995-11-22 EP disclosed
US-5455265-A For mammals; skin disorders, cancer, inflammatory disease, cardiovascular diorders, autoimmune diseases and others ALLERGAN, INC. (US) 1995-10-03 US disclosed
WO-1994017796-A1 THERAPEUTIC USE OF COMPOUNDS HAVING SELECTIVE AGONIST-LIKE ACTIVITY ON RXR RETINOID RECEPTORS ALLERGAN, INC. (US) 1994-08-18 WO disclosed
US-5324840-A Skin disorders ALLERGAN, INC. (US) 1994-06-28 US disclosed