SCHEMBL7223369

SCHEMBL7223369

CCn1nnc([C@H]2O[C@@H](n3cnc4c(N[C@H](CO)Cc5ccccc5)nc(NCCc5cn(C)cn5)nc43)[C@H](O)[C@@H]2OC(C)=O)n1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.56
ADORA3 P0DMS8 16/20 0.56
ADORA1 P30542 11/20 0.56
ADORA2B P29275 9/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7463425 0.91 ADORA2A (0.67) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7231463 0.91 ADORA3 (0.48) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7231458 0.87 ADORA3 (0.48) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7224896 0.85 ADORA3 (0.44) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7459130 0.85 ADORA2A (0.57) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7224384 0.84 ADORA3 (0.53) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7454689 0.84 ADORA2A (0.57) ADORA2AADORA3ADORA1ADORA2B
Acetic Acid SCHEMBL7231454 0.84 ADORA3 (0.52) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7222870 0.82 ADORA2A (0.48) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7229729 0.82 ADORA2A (0.48) ADORA2AADORA3ADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6528494-B2 Antiinflammatory agents COX BRIAN (GB) 2003-03-04 US disclosed
EP-0948509-B1 2-(PURIN-9-YL)-TETRAHYDROFURAN-3,4-DIOL DERIVATIVES GLAXO GROUP LTD (GB) 2002-10-16 EP disclosed
US-6426337-B1 ANTIINFLAMMATORY AGENTS SMITHKLINE BEECHAM CORPORATION 2002-07-30 US disclosed