SCHEMBL7224757

SCHEMBL7224757

CCOC(=O)c1ccc(C=Cc2ccc(CO[Si](C)(C)C(C)(C)C)c(C(C)C)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.41
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
CA14 Q9ULX7 2/20 0.39
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
RAB9A P51151 5/20 0.36
NPC1 O15118 4/20 0.36
MAPT P10636 4/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 2/20 0.36
CYP1A2 P05177 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSP90AA1 P07900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224755 0.84 CA12 (0.39) CA12CA1CA2CA7CA9
SCHEMBL5735225 0.84 ACACB (0.40) CA12CA1CA2CA7CA9
SCHEMBL7224760 0.73 CA12 (0.37) CA12CA1CA2CA7CA9
SCHEMBL24844876 0.73 CA12 (0.52) BACE1CA12CA1CA2CA7
SCHEMBL6619617 0.72 CA12 (0.41) CA12CA1CA2CA7CA9
SCHEMBL9717146 0.71 CA1 (0.66) CA12CA1CA2CA7CA9
SCHEMBL9717141 0.71 CA1 (0.66) CA12CA1CA2CA7CA9
SCHEMBL10618582 0.71 CA1 (0.66) CA12CA1CA2CA7CA9
SCHEMBL13582672 0.69 BACE1 (0.51) BACE1CA12CA1CA2CA7
SCHEMBL13582674 0.69 BACE1 (0.51) BACE1CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6531599-B2 RAI=retinoic acid inducible; for example, 4-((8-cyclopropyl-3,4-dihydro-4,4-dimethylspiro(2H-1-benzopyran-2,1' -cyclopropane)-6-yl) ethynyl)-2-fluoro-benzoic acid; use treating diseases responsive to retinoids ALLERGAN SALES, INC. 2003-03-11 US disclosed