SCHEMBL7224755

SCHEMBL7224755

C=C(c1ccc(C(=O)OCC)cc1)c1ccc(CO[Si](C)(C)C(C)(C)C)c(C(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA7 P43166 3/20 0.39
CA9 Q16790 3/20 0.39
CA14 Q9ULX7 3/20 0.39
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
RAB9A P51151 5/20 0.36
CYP1A2 P05177 3/20 0.36
LMNA P02545 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAOA P21397 1/20 0.36
MAPT P10636 5/20 0.35
NPC1 O15118 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
ALDH1A1 P00352 4/20 0.34
HPGD P15428 3/20 0.34
HTT P42858 3/20 0.34
HSP90AA1 P07900 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224757 0.84 BACE1 (0.41) CA12CA1CA2CA7CA9
SCHEMBL5735225 0.84 ACACB (0.40) CA12CA1CA2CA7CA9
SCHEMBL6619617 0.73 CA12 (0.41) CA12CA1CA2CA7CA9
SCHEMBL31075303 0.70 NQO2 (0.37) CA12CA1CA2CA7CA9
SCHEMBL31075219 0.69 GRM2 (0.44) CYP1A2CYP3A4MAPTSMN1; SMN2CYP2C9
SCHEMBL14641532 0.69 CA12 (0.50) CA12CA1CA2CA7CA9
SCHEMBL23066425 0.67 ESR1 (0.47) CA12CA1CA2CA7CA9
SCHEMBL1018742 0.67 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL17544510 0.67 CA12 (0.44) CA12CA1CA2CA7CA9
SCHEMBL16621371 0.67 ALDH1A1 (0.46) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6531599-B2 RAI=retinoic acid inducible; for example, 4-((8-cyclopropyl-3,4-dihydro-4,4-dimethylspiro(2H-1-benzopyran-2,1' -cyclopropane)-6-yl) ethynyl)-2-fluoro-benzoic acid; use treating diseases responsive to retinoids ALLERGAN SALES, INC. 2003-03-11 US disclosed