SCHEMBL7225664

SCHEMBL7225664

Cc1ccccc1-c1ccc(C(=O)N[C@@H]2C[C@H]3CC[C@@H]2N3)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.48
CHRNA7 P36544 10/20 0.47
MAPK11 Q15759 3/20 0.43
MAPK14 Q16539 3/20 0.43
MAPK13 O15264 1/20 0.43
MAPK12 P53778 1/20 0.43
HTR3E A5X5Y0 5/20 0.41
HTR3B O95264 5/20 0.41
HTR3A P46098 5/20 0.41
HTR3D Q70Z44 5/20 0.41
HTR3C Q8WXA8 5/20 0.41
S1PR2 O95136 1/20 0.40
S1PR4 O95977 1/20 0.40
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39
DYRK1A Q13627 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
MCHR1 Q99705 1/20 0.38
KCNH2 Q12809 1/20 0.37
SCN5A Q14524 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223518 0.89 CHRNA7 (0.60) CHRNA7MAPK11MAPK14MAPK13MAPK12
Hydrochloric Acid SCHEMBL7226319 0.88 CHRNA7 (0.59) CHRNA7MAPK11MAPK14MAPK13MAPK12
SCHEMBL7225752 0.88 CHRNA7 (0.45) HPGDCHRNA7HTR3EHTR3BHTR3A
SCHEMBL7223890 0.87 CHRNA7 (0.43) HPGDCHRNA7MAPK11MAPK14MAPK13
SCHEMBL7225837 0.87 CHRNA7 (0.44) HPGDCHRNA7HTR3EHTR3BHTR3A
SCHEMBL7232275 0.86 CHRNA7 (0.62) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7230420 0.85 CHRNA7 (0.42) HPGDCHRNA7MAPK11MAPK14MAPK13
SCHEMBL7226736 0.85 DYRK1A (0.44) HPGDCHRNA7MAPK11MAPK14MAPK13
SCHEMBL7232588 0.85 HPGD (0.50) HPGDCHRNA7HTR3EHTR3BHTR3A
SCHEMBL7223981 0.84 CHRNA7 (0.42) HPGDCHRNA7MAPK11MAPK14MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed