SCHEMBL7230437

SCHEMBL7230437

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(-c2cc(F)cc(F)c2)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 1/20 0.42
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SLC6A3 Q01959 3/20 0.38
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
POLB P06746 1/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
CHRNA1 P02708 1/20 0.37
CHRNG P07510 1/20 0.37
ITGA5 P08648 1/20 0.37
CHRNB1 P11230 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7075352 0.90 NR4A1 (0.50) SLC9A1NPC1RAB9AALDH1A1KDM4E
SCHEMBL7072340 0.90 PTPN1 (0.46) SLC9A1NPC1RAB9AL3MBTL1SLC6A3
Hydrochloric Acid SCHEMBL7072319 0.89 NR4A1 (0.49) SLC9A1NPC1RAB9AALDH1A1KDM4E
Hydrochloric Acid SCHEMBL7074856 0.89 PTPN1 (0.46) SLC9A1NPC1RAB9AL3MBTL1SLC6A3
SCHEMBL7225315 0.89 AKT1 (0.39) NPC1RAB9AL3MBTL1SLC6A3ALDH1A1
SCHEMBL7224342 0.87 NPC1 (0.42) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7224388 0.87 NPC1 (0.46) SLC9A1NPC1RAB9AL3MBTL1SLC6A3
SCHEMBL7223707 0.85 NPC1 (0.38) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL375394 0.85 NPC1 (0.44) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7074460 0.85 NPC1 (0.44) NPC1RAB9AL3MBTL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed