SCHEMBL7224388

SCHEMBL7224388

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(-c2cc(Cl)cc(Cl)c2)o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
AKT1 P31749 4/20 0.42
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 3/20 0.42
LMNA P02545 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MAPT P10636 2/20 0.42
SLC9A1 P19634 1/20 0.42
HPGD P15428 2/20 0.40
GPR55 Q9Y2T6 1/20 0.40
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
S1PR4 O95977 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7225482 0.90 ALDH1A1 (0.54) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7226254 0.90 NPC1 (0.59) NPC1RAB9AL3MBTL1AKT1ALDH1A1
Hydrochloric Acid SCHEMBL7231981 0.89 NPC1 (0.58) NPC1RAB9AL3MBTL1AKT1ALDH1A1
SCHEMBL7232165 0.89 AKT1 (0.43) NPC1RAB9AL3MBTL1AKT1ALDH1A1
SCHEMBL7234436 0.87 NPC1 (0.45) NPC1RAB9AL3MBTL1AKT1ALDH1A1
SCHEMBL7230437 0.87 SLC9A1 (0.42) NPC1RAB9AL3MBTL1AKT1ALDH1A1
SCHEMBL7074460 0.85 NPC1 (0.44) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL375394 0.85 NPC1 (0.44) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL7224342 0.85 NPC1 (0.42) NPC1RAB9AL3MBTL1AKT1ALDH1A1
SCHEMBL7223159 0.84 RAB9A (0.39) NPC1RAB9AL3MBTL1AKT1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed