SCHEMBL7231502

SCHEMBL7231502

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(-c2cccnc2)o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.46
CHRNA4 P43681 3/20 0.46
CHRNA7 P36544 2/20 0.46
NPC1 O15118 1/20 0.42
POLB P06746 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 2/20 0.40
MAPT P10636 2/20 0.40
CHRNA3 P32297 1/20 0.40
AKT1 P31749 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PTPN22 Q9Y2R2 1/20 0.38
CDK2 P24941 1/20 0.38
KDR P35968 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223139 0.87 NPC1 (0.42) CHRNB2CHRNA4CHRNA7NPC1POLB
SCHEMBL375394 0.87 NPC1 (0.44) CHRNB2CHRNA4CHRNA7NPC1POLB
SCHEMBL7074460 0.87 NPC1 (0.44) CHRNB2CHRNA4CHRNA7NPC1POLB
Hydrochloric Acid SCHEMBL7075781 0.86 NPC1 (0.43) CHRNB2CHRNA4CHRNA7NPC1POLB
SCHEMBL7232969 0.84 FAAH (0.42) CHRNB2CHRNA4NPC1RAB9AALDH1A1
SCHEMBL7232165 0.84 AKT1 (0.43) NPC1POLBMAPK1RAB9AALDH1A1
SCHEMBL7225315 0.84 AKT1 (0.39) NPC1POLBRAB9AALDH1A1KDM4E
SCHEMBL7226285 0.83 NPC1 (0.44) CHRNB2CHRNA4CHRNA7NPC1POLB
SCHEMBL7224267 0.83 NPC1 (0.39) CHRNB2CHRNA4NPC1POLBRAB9A
SCHEMBL7224791 0.82 NPC1 (0.44) NPC1POLBRAB9AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed