SCHEMBL7233992

SCHEMBL7233992

Cc1cc(Nc2ncnc3ccc(OC(=O)C#CCCCCN4CCOCC4)cc23)ccc1Cc1ccsc1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 8/20 0.47
EGFR P00533 15/20 0.45
ERBB4 Q15303 4/20 0.45
SRC P12931 3/20 0.41
KDR P35968 3/20 0.41
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7233687 0.80 AURKA (0.51) ERBB2EGFRERBB4SRCKDR
SCHEMBL7242049 0.80 EGFR (0.61) ERBB2EGFRERBB4SRCKDR
SCHEMBL7244702 0.80 EGFR (0.48) ERBB2EGFRERBB4SRCKDR
SCHEMBL7121729 0.79 EGFR (0.49) ERBB2EGFRERBB4SRC
SCHEMBL7125412 0.77 EGFR (0.48) ERBB2EGFRERBB4SRC
SCHEMBL7242855 0.76 EGFR (0.65) ERBB2EGFRERBB4
SCHEMBL7242169 0.74 ERBB2 (0.51) ERBB2EGFRERBB4KDR
SCHEMBL7117608 0.72 EGFR (0.54) ERBB2EGFRERBB4
SCHEMBL7130805 0.72 AURKA (0.44) ERBB2EGFRERBB4SRCKDR
SCHEMBL7237483 0.71 EGFR (0.63) ERBB2EGFRERBB4SRCKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127374-A AN ENZYME INHIBITOR FOR TREATING CANCER, RESTENOSIS, ATHEROSCLEROSIS, ENDOMETRIOSIS AND PSORIASIS WARNER-LAMBERT COMPANY (US) 2000-10-03 US claimed
US-6562818-B1 For treating cancer, atherosclerosis, restenosis, endometriosis, and psoriasis WARNER-LAMBERT COMPANY 2003-05-13 US disclosed
US-6127374-A AN ENZYME INHIBITOR FOR TREATING CANCER, RESTENOSIS, ATHEROSCLEROSIS, ENDOMETRIOSIS AND PSORIASIS WARNER-LAMBERT COMPANY (US) 2000-10-03 US disclosed