SCHEMBL7235666

SCHEMBL7235666

COc1ccc(OC)c(-c2ccc(CC(N)C(=O)O)cc2)c1

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TPH1 P17752 15/20 0.69
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
HPGD P15428 1/20 0.50
PPARG P37231 1/20 0.50
PPARA Q07869 1/20 0.50
LDHA P00338 1/20 0.49
SLC9A1 P19634 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6528925 0.92 TPH1 (0.69) TPH1PPARGLDHA
SCHEMBL2000541 0.85 PPARG (0.55) TPH1PPARGPPARALDHA
SCHEMBL30040624 0.84 TPH1 (0.54) TPH1PPARGPPARALDHA
SCHEMBL2000467 0.84 TPH1 (0.54) TPH1PPARGPPARALDHA
SCHEMBL429637 0.84 TPH1 (0.54) TPH1PPARGPPARALDHA
SCHEMBL6168594 0.83 TPH1 (0.68) TPH1PPARGPPARALDHA
SCHEMBL5213839 0.83 PPARG (0.63) TPH1PPARGPPARA
SCHEMBL7227938 0.83 PPARG (0.63) TPH1PPARGPPARA
SCHEMBL31398354 0.83 PPARG (0.63) TPH1PPARGPPARA
SCHEMBL29810055 0.82 TPH1 (1.00) TPH1ALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6645939-B1 Very late antigen-4 (VLA) integrin antagonists; antiallergens, antiasthmatics, and antiinflammatory agents; multiple sclerosis, autoimmune disease treatment MERCK & CO., INC. 2003-11-11 US disclosed