SCHEMBL723573

SCHEMBL723573

CC(=O)[C@](O)(C(=O)Br)[C@@H](O)[C@@H](O)[C@H](O)CO

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PDE4A P27815 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
USP2 O75604 1/20 0.33
SLCO1B1 Q9Y6L6 1/20 0.33
KDM4E B2RXH2 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL941684 1.00 LMNA (0.36) LMNAL3MBTL1PDE4ATDP1USP2
SCHEMBL1419602 1.00 LMNA (0.36) LMNAL3MBTL1PDE4ATDP1USP2
SCHEMBL27522036 1.00 LMNA (0.36) LMNAL3MBTL1PDE4ATDP1USP2
SCHEMBL4880937 0.89
SCHEMBL1785079 0.89
SCHEMBL1783279 0.89
SCHEMBL15846054 0.84 LMNA (0.34) LMNAL3MBTL1PDE4ATDP1USP2
SCHEMBL16798768 0.83 PDE4A (0.41) LMNAL3MBTL1PDE4ATDP1USP2
SCHEMBL29162767 0.83 PDE4A (0.41) LMNAL3MBTL1PDE4ATDP1USP2
SCHEMBL5859311 0.83 PDE4A (0.41) LMNAL3MBTL1PDE4ATDP1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 229 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0465998-B1 Beta-galactosidase substrate for CEDIA assays BOEHRINGER MANNHEIM GMBH (DE) 1996-03-06 EP claimed
EP-0310014-B1 Chromogene substrate BEHRINGWERKE AG (DE) 1995-06-21 EP claimed
US-5254677-A β-galactosidase substrates for cedia BOEHRINGER MANNHEIM GMBH (DE) 1993-10-19 US claimed
EP-0465998-A1 Beta-galactosidase substrate for CEDIA assays Roche Diagnostics GmbH (DE) 1992-01-15 EP claimed
US-5077200-A Detection of hydrolyzing enzymes BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1991-12-31 US claimed
JP-1294698-A None JP disclosed
JP-54041863-A None JP disclosed
JP-1115962-A None JP disclosed
JP-4253991-A None JP disclosed
EP-4651911-A1 NEW SENESCENCE TRACER GENERATION Eberhard Karls Universität Tübingen, Medizinische Fakultät (DE) 2025-11-26 EP disclosed
WO-2024189080-A1 NEW SENESCENCE TRACER GENERATION EBERHARD KARLS UNIVERSITAET TUEBINGEN MEDIZINISCHE FAKULTAET (DE) 2024-09-19 WO disclosed
CN-110546154-B Fluorogenic substrates for glycosidases and related detection methods 里昂师范大学 2024-04-05 CN disclosed
US-4281061-A DETECTABLE SIGNAL FROM FLUORESCENT DYE OR LABELED ENZYME SYVA COMPANY (US) 1981-07-28 US disclosed
US-4268663-A COMPRISING A POLYSACCHARIDE SUPPORT, AN AMINE-CONTAINING SPACER ARM, AND A CHROMOGEN ENZYMATICALLY LABILE-LINKED TO A MONOSACCHARIDE; IMMUNOASSAY SYVA COMPANY (US) 1981-05-19 US disclosed
EP-0018731-A1 Macromolecular glycosidase substrates SYVA COMPANY (US) 1980-11-12 EP disclosed
US-4232150-A COMPLEMENT INHIBITORS AMERICAN CYANAMID COMPANY (US) 1980-11-04 US disclosed
US-4221907-A COMPLEMENT INHIBITORS AMERICAN CYANAMID COMPANY (US) 1980-09-09 US disclosed
JP-S5441863-A PRODUCTION OF STEVIOSIDE ANALOGS TAKASAGO CORP 1979-04-03 JP disclosed
US-4038270-A CONDENSING MENTHOL WITH A SUGAR TOYO HAKKA KOBYO KABUSHIKI KAISHA (JA) 1977-07-26 US disclosed
US-3988482-A Menthol glycoside, process for preparing the same and method for releasing menthol therefrom TOYO HAKKA KOGYO KABUSHIKI KAISHA (JA) 1976-10-26 US disclosed