SCHEMBL7235877

SCHEMBL7235877

CC(C)(C)OC(=O)NC(Cc1ccc(O)cc1)C(=O)OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 5/20 0.63
CTSK P43235 4/20 0.63
CTSL P07711 2/20 0.59
CTSB P07858 2/20 0.59
PPARA Q07869 2/20 0.58
ACE P12821 1/20 0.57
KLK5 Q9Y337 1/20 0.55
MAPT P10636 2/20 0.53
POLB P06746 1/20 0.53
MAPK1 P28482 1/20 0.53
KDM4E B2RXH2 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
PPARG P37231 1/20 0.53
ATM Q13315 1/20 0.52
TACR1 P25103 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1486267 1.00 CTSS (0.63) CTSSCTSKCTSLCTSBPPARA
SCHEMBL16163459 1.00 CTSS (0.63) CTSSCTSKCTSLCTSBPPARA
SCHEMBL85543 0.95 CTSS (0.64) CTSSCTSKCTSLCTSBPPARA
SCHEMBL22404737 0.95 CTSS (0.64) CTSSCTSKCTSLCTSBPPARA
SCHEMBL3355326 0.95 CTSS (0.64) CTSSCTSKCTSLCTSBPPARA
SCHEMBL7409385 0.93 CTSS (0.65) CTSSCTSKCTSLCTSBPPARA
SCHEMBL7409389 0.93 CTSS (0.65) CTSSCTSKCTSLCTSBPPARA
SCHEMBL23729806 0.92 CTSS (0.58) CTSSCTSKCTSLCTSBPPARA
SCHEMBL24942151 0.92 CTSS (0.58) CTSSCTSKCTSLCTSBPPARA
SCHEMBL16355883 0.92 CTSS (0.58) CTSSCTSKCTSLCTSBPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
CN-1057760-C Amino acid-substituted benzoylguanidines, a process for their preparation, their use as a medicament or diagnostic agent and a medicament containing them HOECHST AG (DE) 2000-10-25 CN disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
US-5631293-A CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1997-05-20 US disclosed
CN-1138321-A 1, 3-dialkyl urea derivative with hydrocarbon group SANTAN PHARMACEUTICAL CO LTD (JP) 1996-12-18 CN disclosed
CN-1127749-A Amino acid-substituted benzoylguanidines, a process for their preparation, their use as a medicament or diagnostic agent and a medicament containing them HOECHST AG (DE) 1996-07-31 CN disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed