SCHEMBL7236140

SCHEMBL7236140

CC(C)(C)[Si](C)(C)Oc1ccc(-c2ccc([C@H](N)CC(=O)O)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PREP P48147 4/20 0.43
FFAR1 O14842 11/20 0.41
TPH1 P17752 1/20 0.39
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7236266 0.96 PREP (0.40) PREPFFAR1TPH1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL7236572 0.95 PREP (0.39) PREPFFAR1TPH1KMT2ASMN1; SMN2
SCHEMBL7237737 0.83 PREP (0.41) PREPKMT2ACA12CA1CA9
SCHEMBL7455145 0.83 PREP (0.41) PREPKMT2ACA12CA1CA9
SCHEMBL7236135 0.82 PREP (0.40) PREP
SCHEMBL10317188 0.81 PREP (0.41) PREPFFAR1KMT2ASMN1; SMN2CA12
SCHEMBL5624168 0.81 KDM4E (0.40) PREPCA12CA1CA9
SCHEMBL5624172 0.81 KDM4E (0.40) PREPCA12CA1CA9
SCHEMBL10317583 0.76 FFAR1 (0.55) FFAR1
SCHEMBL27582399 0.76 KMT2A (0.43) FFAR1TPH1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6645939-B1 Very late antigen-4 (VLA) integrin antagonists; antiallergens, antiasthmatics, and antiinflammatory agents; multiple sclerosis, autoimmune disease treatment MERCK & CO., INC. 2003-11-11 US disclosed