SCHEMBL7455145

SCHEMBL7455145

COC(=O)CC(N)c1ccc(O[Si](C)(C)C(C)(C)C)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PREP P48147 4/20 0.41
CA12 O43570 3/20 0.35
CA1 P00915 3/20 0.35
CA9 Q16790 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MAPT P10636 3/20 0.35
RAB9A P51151 1/20 0.35
HTT P42858 3/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ADRB3 P13945 1/20 0.33
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7237737 1.00 PREP (0.41) PREPCA12CA1CA9CYP1A2
SCHEMBL5624168 0.87 KDM4E (0.40) PREPCA12CA1CA9MAPT
SCHEMBL5624172 0.87 KDM4E (0.40) PREPCA12CA1CA9MAPT
SCHEMBL7236266 0.86 PREP (0.40) PREPCA12CA1CA9CYP1A2
Hydrochloric Acid SCHEMBL7236572 0.85 PREP (0.39) PREPCA12CA1CA9KMT2A
SCHEMBL1508406 0.85 PREP (0.42) PREPCA12CA1CA9NPSR1
SCHEMBL7236140 0.83 PREP (0.43) PREPCA12CA1CA9KMT2A
SCHEMBL1508330 0.81 FFAR1 (0.42) PREP
SCHEMBL17493569 0.80 FFAR1 (0.39) PREPCA12CA1CA9NPSR1
SCHEMBL17493578 0.80 FFAR1 (0.39) PREPCA12CA1CA9NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1034164-A4 SUBSTITUTED BETA-ALANINE DERIVATIVES AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2001-07-11 EP disclosed
EP-1034164-A1 SUBSTITUTED BETA-ALANINE DERIVATIVES AS CELL ADHESION INHIBITORS Merck & Co., Inc. (US) 2000-09-13 EP disclosed
WO-1999026921-A1 SUBSTITUTED β-ALANINE DERIVATIVES AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-06-03 WO disclosed