SCHEMBL7239268

SCHEMBL7239268

CN(C)CC(O)COc1ccc(Nc2ncc(CO)c(Nc3ccccc3)n2)cc1

nearest known ligand 0.78

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.78
CDK2 P24941 17/20 0.78
CDK1 P06493 1/20 0.50
CCNE1 P24864 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7236132 0.89 CDK4 (0.72) CDK4CDK2CDK1CCNE1
SCHEMBL6644644 0.89 CDK4 (0.75) CDK4CDK2CDK1CCNE1
Hydrochloric Acid SCHEMBL7232203 0.88 CDK4 (0.73) CDK4CDK2CDK1CCNE1
SCHEMBL7238750 0.88 CDK4 (0.72) CDK4CDK2CDK1CCNE1
SCHEMBL29644990 0.87 CDK4 (1.00) CDK4CDK2
SCHEMBL6645907 0.87 CDK4 (0.80) CDK4CDK2CDK1CCNE1
SCHEMBL29644986 0.87 CDK4 (1.00) CDK4CDK2
SCHEMBL5581900 0.87 CDK4 (1.00) CDK4CDK2
SCHEMBL14632119 0.87 CDK4 (1.00) CDK4CDK2CCNE1
SCHEMBL6643501 0.86 CDK4 (0.69) CDK4CDK2CDK1CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6593326-B1 Useful as anti-cancer agents; and processes for their manufacture and pharmaceutical compositions containing them are described. Apoptotic effect in a warm-blooded animal such as man. ASTRAZENECA AB (SE) 2003-07-15 US disclosed