SCHEMBL7239455

SCHEMBL7239455

COc1ccccc1CN1CCN(c2ncccc2C(=O)NC(C=O)Cc2ccccc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 7/20 0.49
CTSS P25774 1/20 0.49
GPR6 P46095 1/20 0.46
KDM4E B2RXH2 3/20 0.46
ALOX15 P16050 1/20 0.46
EPHX2 P34913 1/20 0.45
BCHE P06276 2/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CXCR4 P61073 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7235830 0.88 CAPN1 (0.56) CAPN1CTSSBCHETSHR
SCHEMBL7238926 0.87 CAPN1 (0.49) CAPN1CTSSGPR6BCHEMAPT
SCHEMBL7242368 0.87 CAPN1 (0.49) CAPN1CTSSGPR6KDM4EALOX15
SCHEMBL7241474 0.87 CAPN1 (0.51) CAPN1CTSSGPR6KDM4EALDH1A1
SCHEMBL7242371 0.85 GPR6 (0.48) CAPN1CTSSGPR6KDM4EALOX15
SCHEMBL7243236 0.85 L3MBTL1 (0.49) CAPN1CTSSGPR6MAPTTSHR
SCHEMBL7238735 0.84 CAPN1 (0.53) CAPN1CTSSTSHRMEN1KMT2A
SCHEMBL7242851 0.83 CHIA (0.58) CAPN1CTSSTSHR
SCHEMBL7243833 0.82 CAPN1 (0.69) CAPN1CTSSKDM4EALDH1A1MAPT
SCHEMBL7232336 0.82 CAPN1 (0.58) CAPN1CTSSALDH1A1TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562827-B1 For the treatment of diseases in which increased calpain activity occurs such as neurodegenerative diseases or neuronal damage are caused by ischemia, trauma or mass hemorrhages ABBOTT LABORATORIES 2003-05-13 US disclosed