SCHEMBL7243743

SCHEMBL7243743

COc1ccc(S(=O)(=O)Nc2cc(C(=N)N)sc2SC)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.51
NFE2L2 Q16236 1/20 0.51
C1S P09871 6/20 0.51
ALDH1A1 P00352 3/20 0.50
TP53 P04637 1/20 0.50
LMNA P02545 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
HTT P42858 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
TSHR P16473 1/20 0.49
CYP2C9 P11712 1/20 0.47
CA12 O43570 1/20 0.47
CA9 Q16790 1/20 0.47
PLAU P00749 1/20 0.47
FFAR4 Q5NUL3 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7242045 0.87 C1S (0.59) KEAP1NFE2L2C1SALDH1A1LMNA
SCHEMBL6926242 0.83 C1S (0.56) C1SALDH1A1PLAU
SCHEMBL7246060 0.82 CCR2 (0.52) C1SPLAU
SCHEMBL7245020 0.82 C1S (0.50) C1SPLAU
SCHEMBL7242120 0.82 C1S (0.65) C1SALDH1A1SMN1; SMN2PLAU
SCHEMBL6928674 0.82 C1S (0.69) C1SMEN1KMT2APLAU
SCHEMBL6927266 0.81 C1S (0.63) C1S
SCHEMBL6925664 0.81 C1S (0.62) C1SPLAU
SCHEMBL6925869 0.80 C1S (0.54) C1SPLAU
SCHEMBL7241070 0.80 C1S (0.48) C1SPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562840-B1 Non-peptidic inhibitors of proteolytic enzymes such as urokinase 3-DIMENSIONAL PHARMACEUTICALS, INC. 2003-05-13 US claimed