SCHEMBL7244100

SCHEMBL7244100

Fc1ccc(-c2n[nH]cc2-c2ccnc(NCCC3CCCCN3C3CCNCC3)c2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.37
MAPK9 P45984 2/20 0.37
EGFR P00533 1/20 0.37
RAF1 P04049 1/20 0.37
ERBB2 P04626 1/20 0.37
MAPK8 P45983 1/20 0.37
MAPK14 Q16539 18/20 0.36
MAPK13 O15264 3/20 0.36
MAPK12 P53778 3/20 0.36
MAPK11 Q15759 3/20 0.36
PRKD3 O94806 2/20 0.34
MAP4K4 O95819 2/20 0.34
PRKACA P17612 2/20 0.34
CSNK1A1 P48729 2/20 0.34
CSNK1D P48730 2/20 0.34
MINK1 Q8N4C8 2/20 0.34
MAP4K5 Q9Y4K4 2/20 0.34
HSPB1 P04792 1/20 0.34
PRKCB P05771 1/20 0.34
PRKCA P17252 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5452474 0.85 MAPK14 (0.39) MAPK14MAPK13MAPK12MAPK11
SCHEMBL5453721 0.79 MAPK14 (0.50) KDRMAPK9EGFRRAF1ERBB2
SCHEMBL14519560 0.77 HRH3 (0.40) MAPK14MAPK13MAPK12MAPK11
SCHEMBL5447721 0.77 MAP4K4 (0.48) MAPK14MAPK13MAPK12MAPK11MAP4K4
SCHEMBL5463476 0.76 SIGMAR1 (0.40) MAPK14MAPK13MAPK12MAPK11MAP4K4
SCHEMBL5453641 0.76 KDM4E (0.45) MAPK14
SCHEMBL7151203 0.76 MAPK14 (0.52) KDRMAPK9EGFRRAF1ERBB2
SCHEMBL14521999 0.74 MAPK14 (0.54) EGFRMAPK14MAPK13MAPK12MAPK11
SCHEMBL5452518 0.72 MAPK14 (0.56) MAPK14MAPK13MAPK12MAPK11CSNK2A1
SCHEMBL27540765 0.72 MAPK14 (0.41) MAPK14MAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6617324-B1 Phenyl, cyclohexyl and pyridinyl or pyrimidinyl-substituted G. D. SEARLE & COMPANY 2003-09-09 US disclosed