SCHEMBL7248152

SCHEMBL7248152

CCOC(=O)C(=Cc1ccc(F)cc1)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.64
MEN1 O00255 5/20 0.64
KMT2A Q03164 5/20 0.64
LMNA P02545 3/20 0.64
NPSR1 Q6W5P4 3/20 0.64
CYP1A2 P05177 1/20 0.64
CYP2C9 P11712 1/20 0.64
CYP2C19 P33261 1/20 0.64
POLB P06746 1/20 0.54
ALDH1A1 P00352 3/20 0.50
KDM4E B2RXH2 1/20 0.50
HSP90AA1 P07900 1/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 2/20 0.48
NR1H4 Q96RI1 1/20 0.47
AKR1C1 Q04828 2/20 0.47
PTGS2 P35354 1/20 0.47
AKR1C2 P52895 1/20 0.47
AKR1C3 P42330 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7248148 0.94 MEN1 (0.64) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL24704034 0.90 MEN1 (0.70) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL648889 0.90 MEN1 (0.70) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL7527305 0.90 MEN1 (0.70) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL14970302 0.84 KMT2A (0.55) MAPTMEN1KMT2ALMNAALDH1A1
SCHEMBL6934839 0.83 MEN1 (0.57) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL6934835 0.83 MEN1 (0.57) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL3218584 0.79 MAPT (1.00) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL10728016 0.79 ALDH1A1 (0.54) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL6170117 0.79 MEN1 (0.62) MAPTMEN1KMT2ALMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6590102-B1 Hydrogenation of 2-cyano-3-(p-fluorophenyl)glutaric acid diethyl ester in the presence of catalysts to prepare isomer mixtures of ethyl 4-(p-fluorophenyl)-6-oxo-3-piperidine -carboxylate, used as intermediates of paroxetine ASAHI GLASS COMPANY LTD. (JP) 2003-07-08 US disclosed
US-6476228-B1 Process for producing piperidinecarbinols ASAHI GLASS COMPANY LTD. (JP) 2002-11-05 US disclosed
EP-0802185-B1 Process for producing piperidinecarbinols ASAHI GLASS CO LTD (JP) 2001-10-17 EP disclosed
US-6197960-B1 REDUCTION OF CYANOGLUTARIC ACID; CYCLIZATION, ISOMERIZATION ASAHI GLASS COMPANY LTD. (JP) 2001-03-06 US disclosed
EP-0802185-A1 Process for producing piperidinecarbinols ASAHI GLASS COMPANY LTD. (JP) 1997-10-22 EP disclosed