SCHEMBL7248576

SCHEMBL7248576

CCOC(=O)CCCSc1ccc(Br)cc1C=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
PTGDR2 Q9Y5Y4 3/20 0.39
MAPT P10636 5/20 0.38
KMT2A Q03164 4/20 0.38
HPGD P15428 2/20 0.38
CYP3A4 P08684 1/20 0.38
MEN1 O00255 2/20 0.37
S1PR4 O95977 1/20 0.37
LMNA P02545 1/20 0.37
S1PR1 P21453 1/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ERN1 O75460 1/20 0.37
KDM4E B2RXH2 1/20 0.37
GLA P06280 1/20 0.37
POLB P06746 1/20 0.36
PABPC1 P11940 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16334449 0.82 CYP1A2 (0.40) ALDH1A1CYP1A2CYP2C19PTGDR2MAPT
SCHEMBL30350667 0.82 CYP1A2 (0.40) ALDH1A1CYP1A2CYP2C19PTGDR2MAPT
SCHEMBL7246626 0.82 PTGDR2 (0.46) ALDH1A1CYP1A2CYP2C19PTGDR2MAPT
SCHEMBL7253135 0.81 ERN1 (0.46) ALDH1A1HPGDMAPK1ERN1
SCHEMBL7248509 0.79 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP2C19MAPTHPGD
SCHEMBL5550248 0.79 PTGDR2 (0.57) ALDH1A1CYP1A2CYP2C19PTGDR2MAPT
SCHEMBL3459019 0.78 PTGDR2 (0.56) ALDH1A1CYP1A2CYP2C19PTGDR2MAPT
SCHEMBL16146944 0.77 PTGDR2 (0.54) ALDH1A1CYP1A2CYP2C19PTGDR2MAPT
SCHEMBL7541385 0.77 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP2C19PTGDR2MAPT
SCHEMBL15228885 0.76 SMN1; SMN2 (0.47) ALDH1A1CYP1A2CYP2C19PTGDR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6566535-B1 Causing an orthohalogenobenzaldehyde or derivative to react with a propanethiol having an electron-attracting group at its 4- position. TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-05-20 US disclosed
EP-1184381-A1 PROCESSES FOR THE PREPARATION OF 2,3-DIHYDROTHIEPINE DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2002-03-06 EP disclosed