SCHEMBL7253117

SCHEMBL7253117

COC(=O)CCc1c(-c2ccc(O)cc2)[nH]c2nccnc12

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 19/20 0.69
GSK3B P49841 19/20 0.69
CDK1 P06493 18/20 0.69
CCNB2 O95067 17/20 0.69
CCNB1 P14635 17/20 0.69
CCNB3 Q8WWL7 17/20 0.69
CDK5 Q00535 11/20 0.69
CDK5R1 Q15078 10/20 0.69
MAPK8 P45983 3/20 0.66
CDK2 P24941 3/20 0.66
CCNE1 P24864 2/20 0.66
CCNE2 O96020 1/20 0.66
INSR P06213 1/20 0.66
CFTR P13569 1/20 0.66
CCNA2 P20248 1/20 0.66
MAPK3 P27361 1/20 0.66
MAPK1 P28482 1/20 0.66
MAPK9 P45984 1/20 0.66
MAPK10 P53779 1/20 0.66
CCNA1 P78396 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1778932 0.90 GSK3A (0.69) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1778366 0.86 GSK3A (0.70) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1779346 0.86 GSK3A (0.70) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1779469 0.85 GSK3A (0.69) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL7253083 0.82 GSK3A (0.53) GSK3AGSK3BCDK1CCNB2CCNB1
Bromide SCHEMBL490395 0.81 GSK3A (0.97) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL27594653 0.81 GSK3A (0.70) GSK3AGSK3BCDK1CCNB2CCNB1
Aloisine A SCHEMBL80147 0.80 GSK3A (1.00) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777822 0.80 GSK3A (0.72) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777268 0.78 GSK3A (0.69) GSK3AGSK3BCDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003000690-A1 SYNTHESIS OF HETEROCYCLIC COMPOUNDS EMPLOYING MICROWAVE TECHNOLOGY AVENTIS PHARMACEUTICALS INC. (US) 2003-01-03 WO disclosed