SCHEMBL7258103

SCHEMBL7258103

O=C(OC(c1ccccc1)c1ccccc1)c1[c]cccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.51
ESR2 Q92731 1/20 0.51
LMNA P02545 3/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
SRC P12931 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.38
KIF11 P52732 1/20 0.35
CYP2D6 P10635 1/20 0.35
SRD5A2 P31213 1/20 0.35
MAPK1 P28482 1/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7700919 0.83 SRC (0.37) ESR1ESR2LMNAALDH1A1SRC
SCHEMBL11082448 0.83 ESR1 (0.41) ESR1ESR2LMNAALDH1A1KDM4E
SCHEMBL10688255 0.81 KMT2A (0.38) ESR1ESR2LMNAALDH1A1KDM4E
SCHEMBL130469 0.79 PDCD1 (0.47) LMNAALDH1A1KDM4EHPGDTP53
SCHEMBL28752431 0.77 ESR1 (0.59) ESR1ESR2LMNAALDH1A1KDM4E
SCHEMBL7258105 0.74 ESR1 (0.67) ESR1ESR2LMNAALDH1A1KDM4E
SCHEMBL28674746 0.74 ESR1 (0.85) ESR1ESR2LMNAALDH1A1KDM4E
SCHEMBL20483494 0.74 ESR1 (0.79) ESR1ESR2LMNAALDH1A1KDM4E
SCHEMBL28058117 0.74 ESR1 (0.61) ESR1ESR2LMNAALDH1A1KDM4E
SCHEMBL6953946 0.73 MAPT (0.41) LMNAALDH1A1KDM4EHPGDCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003072537-A2 SELECTIVE PROTEIN TYROSINE PHOSPHATATASE INHIBITORS ABBOTT LABORATORIES (US) 2003-09-04 WO disclosed
EP-0005889-B1 PROCESS FOR THE PREPARATION OF BETA-LACTAM DERIVATIVES, THE NOVEL DERIVATIVES SO OBTAINABLE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Technobiotic Ltd. (CH) 1982-06-16 EP disclosed
EP-0005889-A1 Process for the preparation of beta-lactam derivatives, the novel derivatives so obtainable and pharmaceutical compositions containing them Technobiotic Ltd. (CH) 1979-12-12 EP disclosed