SCHEMBL7258149

SCHEMBL7258149

NC(=O)c1cc2c(cc1O)OCO2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.43
RAB9A P51151 5/20 0.43
ADRB2 P07550 3/20 0.41
ADRB1 P08588 3/20 0.41
ADRB3 P13945 3/20 0.41
ADRA1D P25100 3/20 0.41
ADRA1A P35348 3/20 0.41
ADRA1B P35368 3/20 0.41
CYP3A4 P08684 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CASP3 P42574 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
CTNNB1 P35222 1/20 0.40
MAPK8 P45983 1/20 0.40
PARP1 P09874 1/20 0.40
TSHR P16473 1/20 0.39
PI4K2A Q9BTU6 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29828929 0.82 CTNNB1 (0.55) CYP3A4SMN1; SMN2ALDH1A1MAPK1CTNNB1
SCHEMBL5391668 0.82 CTNNB1 (0.55) CYP3A4SMN1; SMN2ALDH1A1MAPK1CTNNB1
SCHEMBL7668928 0.80 MAPT (0.50) NPC1RAB9ACYP3A4SMN1; SMN2CASP3
SCHEMBL773047 0.80 KDM4E (0.51) CYP3A4SMN1; SMN2ALDH1A1MAPK1TSHR
SCHEMBL23643822 0.76 ALDH1A1 (0.44) NPC1RAB9ACYP3A4SMN1; SMN2ALDH1A1
SCHEMBL8569388 0.76 KDM4E (0.54) NPC1RAB9AADRB2ADRB1ADRB3
SCHEMBL28568470 0.76 KDM4E (0.50) NPC1RAB9ACYP3A4SMN1; SMN2ALDH1A1
SCHEMBL2268770 0.75 CYP3A4 (0.56) NPC1RAB9ACYP3A4SMN1; SMN2ALDH1A1
SCHEMBL23511720 0.75 ALDH1A1 (0.52) CYP3A4ALDH1A1MAPK1PARP1TSHR
SCHEMBL24163158 0.73 HPGD (0.58) NPC1RAB9ACYP3A4SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1067935-B1 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) UNIV CALIFORNIA (US) 2003-08-20 EP disclosed
EP-1067935-A4 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) UNIV CALIFORNIA (US) 2001-10-04 EP disclosed
EP-1067935-A1 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) The Regents of the University of California (US) 2001-01-17 EP disclosed
US-6124278-A COGNITION ACTIVATORS FOR LEARNING/MEMORY ENHANCEMENT AND TREATMENT OF BRAIN/PSYCHOLOGICAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2000-09-26 US disclosed
WO-1999051240-A1 ACYLBENZOXAZINES FOR ENHANCING SYNAPTIC RESPONSE(S) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1999-10-14 WO disclosed