SCHEMBL7258795

SCHEMBL7258795

O=C(O)c1nc(N2CCCS2(=O)=O)c2cccnc2c1O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CALCA P06881 7/20 0.69
KDM4E B2RXH2 3/20 0.39
KDM4A O75164 2/20 0.39
EGLN1 Q9GZT9 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
KDM6B O15054 1/20 0.39
KDM6A O15550 1/20 0.39
TET3 O43151 1/20 0.39
KDM4B O94953 1/20 0.39
KDM5C P41229 1/20 0.39
KDM4D Q6B0I6 1/20 0.39
TET2 Q6N021 1/20 0.39
ALKBH5 Q6P6C2 1/20 0.39
TET1 Q8NFU7 1/20 0.39
FTO Q9C0B1 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM2A Q9Y2K7 1/20 0.39
KDM3A Q9Y4C1 1/20 0.39
POLB P06746 1/20 0.37
COMT P21964 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4769028 0.97 CALCA (0.74) CALCAKDM4EKDM4AEGLN1L3MBTL1
SCHEMBL7258799 0.89 CALCA (0.56) CALCAKDM4EKDM4AEGLN1L3MBTL1
SCHEMBL4067727 0.87 CALCA (0.65) CALCAKDM4EL3MBTL1COMT
SCHEMBL4769035 0.85 CALCA (0.60) CALCAKDM4EKDM4AEGLN1L3MBTL1
SCHEMBL4764998 0.84 CALCA (0.54) CALCAKDM4EKDM4AEGLN1L3MBTL1
SCHEMBL968119 0.84 CALCA (0.78) CALCACOMT
SCHEMBL4067964 0.84 CALCA (0.69) CALCAKDM4EL3MBTL1COMT
SCHEMBL4072599 0.83 CALCA (0.68) CALCAKDM4EL3MBTL1COMT
SCHEMBL4765018 0.82 CALCA (0.52) CALCAKDM4EKDM4AEGLN1L3MBTL1
SCHEMBL4060940 0.81 CALCA (0.95) CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003077857-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2003-09-25 WO disclosed