SCHEMBL7260258

SCHEMBL7260258

COC(=O)C(C#N)Cc1ccc(NC(=O)OC(C)(C)C)nc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.42
HDAC1 Q13547 1/20 0.42
GRIN2B Q13224 1/20 0.38
CTSS P25774 7/20 0.38
CTSK P43235 6/20 0.38
LMNA P02545 1/20 0.38
CTSB P07858 2/20 0.37
CTSL P07711 1/20 0.37
FPR1 P21462 1/20 0.37
CYP17A1 P05093 1/20 0.37
MAPK1 P28482 1/20 0.36
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
SYK P43405 1/20 0.35
PTPN1 P18031 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
SCN9A Q15858 1/20 0.35
ATR Q13535 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7257280 0.85 NAMPT (0.46) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL7260124 0.83 NAMPT (0.44) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL31407652 0.82 KLK5 (0.48) NAMPTHDAC1GRIN2BCTSSCTSK
SCHEMBL5076532 0.80 NAMPT (0.47) NAMPTHDAC1GRIN2BCTSSCTSK
SCHEMBL1429937 0.79 HDAC1 (0.47) NAMPTHDAC1GRIN2BCYP17A1MAPK1
SCHEMBL3211479 0.79 HDAC1 (0.47) NAMPTHDAC1GRIN2BCYP17A1MAPK1
SCHEMBL6058751 0.78 NAMPT (0.44) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL2214542 0.77 ITGB3 (0.47) NAMPTHDAC1GRIN2BCTSSCTSK
SCHEMBL7259895 0.77 HDAC1 (0.41) NAMPTHDAC1GRIN2BCTSSCTSK
SCHEMBL13456709 0.77 NAMPT (0.53) NAMPTHDAC1GRIN2BCYP17A1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003013526-A1 ANTICOAGULANT COMPOUNDS MERCK & CO. INC. (US) 2003-02-20 WO disclosed