SCHEMBL7260405

SCHEMBL7260405

Nc1n[nH]c2ccc(-c3ccccc3)nc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.51
GSK3A P49840 1/20 0.51
GSK3B P49841 1/20 0.51
PDPK1 O15530 3/20 0.50
AURKA O14965 2/20 0.50
AURKB Q96GD4 2/20 0.50
TGFBR1 P36897 1/20 0.50
MAP4K1 Q92918 3/20 0.49
KDM4E B2RXH2 2/20 0.44
CYP3A4 P08684 1/20 0.44
GAA P10253 1/20 0.44
MAPK1 P28482 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ASIC3 Q9UHC3 1/20 0.43
KMT2A Q03164 3/20 0.42
AKT2 P31751 1/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 2/20 0.41
RAB9A P51151 1/20 0.41
CYP1A2 P05177 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22744021 0.82 JAK2 (0.47) JAK2PDPK1AURKAAURKBTGFBR1
SCHEMBL29472092 0.82 JAK2 (0.47) JAK2GSK3AGSK3BPDPK1AURKA
SCHEMBL22716353 0.82 JAK2 (0.47) JAK2GSK3AGSK3BPDPK1AURKA
SCHEMBL2036225 0.81 MAP4K1 (0.70) AURKBMAP4K1KDM4EGAAALDH1A1
SCHEMBL30675639 0.74 AURKB (0.51) JAK2GSK3AGSK3BPDPK1AURKA
SCHEMBL13329926 0.74 AURKB (0.51) JAK2GSK3AGSK3BPDPK1AURKA
SCHEMBL3640606 0.74 PDPK1 (0.43) JAK2PDPK1KDM4ECYP3A4GAA
SCHEMBL19994996 0.71 JAK2 (0.47) JAK2PDPK1KDM4ECYP3A4GAA
SCHEMBL29498562 0.71 JAK2 (0.47) JAK2PDPK1KDM4ECYP3A4GAA
SCHEMBL28523916 0.69 KDM4E (0.41) JAK2PDPK1KDM4ECYP3A4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003068773-A1 PYRAZOLOPYRIDINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-08-21 WO disclosed