SCHEMBL7260501

SCHEMBL7260501

COC(=O)c1ccc(CNc2nc(N(C)C)nc3ccc(Cl)cc23)cc1

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 19/20 0.65
TCF7L2 Q9NQB0 19/20 0.65
CNR1 P21554 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7254637 0.87 CNR1 (0.58) CTNNB1TCF7L2CNR1
SCHEMBL7255656 0.79 HRH4 (0.64) CTNNB1TCF7L2
SCHEMBL4168559 0.79 CTNNB1 (1.00) CTNNB1TCF7L2
SCHEMBL4178349 0.79 CTNNB1 (1.00) CTNNB1TCF7L2
SCHEMBL7254554 0.78 CNR1 (0.56) CTNNB1TCF7L2CNR1
SCHEMBL7255329 0.78 HRH4 (0.61) CTNNB1TCF7L2
SCHEMBL4176748 0.77 CTNNB1 (1.00) CTNNB1TCF7L2
SCHEMBL4177162 0.77 CTNNB1 (1.00) CTNNB1TCF7L2
SCHEMBL7254764 0.75 CNR1 (0.57) CTNNB1TCF7L2CNR1
SCHEMBL7258127 0.75 HRH4 (0.60) CTNNB1TCF7L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003055866-A1 QUINAZOLINE AND QUINOLINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO disclosed