SCHEMBL7260601

SCHEMBL7260601

CC(C)COc1cccc(C(N)=O)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.60
NR1H4 Q96RI1 2/20 0.58
SIRT2 Q8IXJ6 1/20 0.56
KAT6A Q92794 2/20 0.54
FOS P01100 1/20 0.53
JUN P05412 1/20 0.53
TNKS O95271 1/20 0.53
PARP15 Q460N3 1/20 0.53
PARP14 Q460N5 1/20 0.53
PARP10 Q53GL7 1/20 0.53
TNKS2 Q9H2K2 1/20 0.53
PARP2 Q9UGN5 1/20 0.53
KMT2A Q03164 3/20 0.50
USP2 O75604 1/20 0.48
TSHR P16473 1/20 0.48
HSD17B1 P14061 1/20 0.48
HSD17B2 P37059 1/20 0.48
OPRK1 P41145 1/20 0.47
MEN1 O00255 1/20 0.46
FABP1 P07148 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16108766 0.87 NR1H4 (0.60) NR1H4SIRT2KAT6AFOSJUN
SCHEMBL1436279 0.85 NR1H4 (0.63) NR1H4KAT6AFOSJUNKMT2A
SCHEMBL931583 0.85 NR1H4 (0.75) NR1H4KAT6AFOSJUNKMT2A
SCHEMBL201949 0.84 NR1H4 (0.60) PARP1NR1H4TNKSPARP15PARP14
SCHEMBL18952331 0.84 PARP1 (0.56) PARP1TNKSPARP15PARP14PARP10
SCHEMBL3248766 0.84 NR1H4 (0.58) NR1H4SIRT2KAT6AFOSJUN
SCHEMBL201166 0.84 PARP1 (0.53) PARP1NR1H4SIRT2TNKSPARP15
SCHEMBL201415 0.83 PARP1 (0.55) PARP1NR1H4TNKSPARP15PARP14
SCHEMBL26049008 0.83 NR1H4 (0.60) NR1H4KAT6AFOSJUNKMT2A
SCHEMBL10431095 0.83 PARP1 (0.54) PARP1TNKSPARP15PARP14PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004000806-A1 AMIDES OF CYCLIC AMINO ACIDS USED AS PDE 4 INHIBITORS ELBION AG (DE) 2003-12-31 WO claimed
WO-2011022393-A2 PHOSPHATIDYLCHOLINE TRANSFER PROTEIN INHIBITORS THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2011-02-24 WO disclosed