SCHEMBL7260688

SCHEMBL7260688

Cc1cc(CBr)cnc1NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LCK P06239 11/20 0.40
AAK1 Q2M2I8 2/20 0.38
CYP17A1 P05093 1/20 0.37
PPARG P37231 1/20 0.36
MAPKAPK2 P49137 2/20 0.36
MAPK14 Q16539 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA9 Q16790 1/20 0.36
AKT1 P31749 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6058971 0.85 STK17B (0.41) AAK1CYP17A1MAPKAPK2MAPK14
SCHEMBL6059191 0.82 MAP4K4 (0.35) LCKAAK1CYP17A1MAPKAPK2MAPK14
SCHEMBL1181471 0.82 AAK1 (0.51) LCKAAK1CA12CA1CA9
SCHEMBL7416577 0.81 LCK (0.45) LCKAAK1MAPKAPK2CA12CA1
SCHEMBL24364156 0.79 MAPKAPK2 (0.40) LCKMAPKAPK2CA12CA1CA9
SCHEMBL7412985 0.79 SYK (0.42) LCKAAK1CYP17A1MAPKAPK2CA12
SCHEMBL30469570 0.79 MAPKAPK2 (0.40) LCKMAPKAPK2CA12CA1CA9
SCHEMBL16786131 0.79 CYP17A1 (0.41) CYP17A1MAPKAPK2CA12CA1AKT1
SCHEMBL15614476 0.77 MAPK1 (0.43) LCKAAK1MAPKAPK2CA12CA1
SCHEMBL7382657 0.76 NR4A1 (0.39) MAPKAPK2CA12CA1AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003013526-A1 ANTICOAGULANT COMPOUNDS MERCK & CO. INC. (US) 2003-02-20 WO disclosed