SCHEMBL24364156

SCHEMBL24364156

Cc1cc(N)cnc1NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 5/20 0.40
MAP4K4 O95819 1/20 0.40
LCK P06239 3/20 0.38
CA1 P00915 2/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
SYK P43405 1/20 0.38
BRD4 O60885 2/20 0.36
ATR Q13535 1/20 0.36
PRMT1 Q99873 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30469570 1.00 MAPKAPK2 (0.40) MAPKAPK2MAP4K4LCKCA1CA12
SCHEMBL7416577 0.85 LCK (0.45) MAPKAPK2LCKCA1CA12CA9
SCHEMBL6517445 0.84 MAPKAPK2 (0.40) MAPKAPK2MAP4K4LCKCA1SYK
SCHEMBL31430396 0.83 MAPKAPK2 (0.41) MAPKAPK2MAP4K4CA1SYKATR
SCHEMBL29477633 0.83 ALDH1A1 (0.40) MAPKAPK2MAP4K4CA1SYKATR
SCHEMBL24367667 0.83 ALDH1A1 (0.40) MAPKAPK2MAP4K4CA1SYKATR
SCHEMBL24364867 0.83 MAPKAPK2 (0.41) MAPKAPK2MAP4K4CA1SYKATR
SCHEMBL7412985 0.82 SYK (0.42) MAPKAPK2LCKCA1CA12CA9
SCHEMBL1181471 0.82 AAK1 (0.51) LCKCA1CA12CA9ATR
SCHEMBL24366932 0.82 LMNA (0.40) MAPKAPK2MAP4K4SYKATRPRMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240228478-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2024-07-11 US disclosed
US-20240228478-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2024-07-11 US disclosed
CN-116568677-A piperidin-1-yl-N-pyridin-3-yl-2-oxoacetamide derivatives useful for the treatment of MTAP deficiency and/or MTA accumulating cancers 探戈医药股份有限公司 2023-08-08 CN disclosed
US-20220127256-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2022-04-28 US disclosed
CN-101808996-A Nicotinamide derivatives, their preparation and their use in therapeutics SANOFI AVENTIS 2010-08-18 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220127256-A1 COMPOUNDS AND METHODS OF USE F12, C1R, ABCG2 MAPKAPK2 4853/4885MAP4K4 4660/4885LCK 3675/4885
US-20240228478-A1 COMPOUNDS AND METHODS OF USE F12, C1R, ABCG2 MAPKAPK2 4853/4885MAP4K4 4660/4885LCK 3675/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.