SCHEMBL7262571

SCHEMBL7262571

COC(=O)c1nc(N2CCCS2(O)O)c2cccnc2c1O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CALCA P06881 6/20 0.53
KDM4E B2RXH2 3/20 0.43
TP53 P04637 2/20 0.36
ALOX15 P16050 2/20 0.36
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
USP2 O75604 1/20 0.36
ALOX12 P18054 1/20 0.36
HTT P42858 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
COMT P21964 1/20 0.35
GAA P10253 1/20 0.35
PSMD14 O00487 1/20 0.34
EGLN1 Q9GZT9 1/20 0.34
MAP2K1 Q02750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4067974 0.97 CALCA (0.56) CALCAKDM4ETP53ALOX15MAPT
SCHEMBL4067727 0.90 CALCA (0.65) CALCAKDM4ETP53ALOX15MAPT
SCHEMBL7258799 0.87 CALCA (0.56) CALCAKDM4ETP53ALOX15L3MBTL1
SCHEMBL4067964 0.87 CALCA (0.69) CALCAKDM4ETP53ALOX15MAPT
SCHEMBL4762094 0.87 CALCA (0.50) CALCAKDM4ETP53ALOX15MAPT
SCHEMBL4072599 0.86 CALCA (0.68) CALCAKDM4ETP53ALOX15MAPT
SCHEMBL4762076 0.84 CALCA (0.52) CALCAKDM4ETP53ALOX15MAPT
SCHEMBL4769035 0.84 CALCA (0.60) CALCAKDM4ETP53ALOX15MAPT
SCHEMBL4064836 0.83 CALCA (0.46) CALCAKDM4ETP53ALOX15MAPT
SCHEMBL968122 0.82 CALCA (0.64) CALCAKDM4ETP53ALOX15MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003077857-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2003-09-25 WO disclosed