SCHEMBL7265907

SCHEMBL7265907

NC(=O)c1nnn(Cc2ccc(C(=O)c3ccc(Cl)cc3)cc2)c1N

nearest known ligand 0.80

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.80
GALR3 O60755 1/20 0.80
CYP3A4 P08684 1/20 0.80
CYP2C9 P11712 1/20 0.80
NR2F2 P24468 1/20 0.80
HIF1A Q16665 1/20 0.80
HTT P42858 1/20 0.55
HPGD P15428 1/20 0.53
MAPT P10636 5/20 0.53
TSHR P16473 2/20 0.51
KMT2A Q03164 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
CYP1A2 P05177 1/20 0.48
ALOX15 P16050 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7265939 0.90 SMN1; SMN2 (0.72) SMN1; SMN2GALR3CYP3A4CYP2C9NR2F2
SCHEMBL10409575 0.90 SMN1; SMN2 (0.65) SMN1; SMN2GALR3CYP3A4CYP2C9NR2F2
Carboxyamidotriazole SCHEMBL18866 0.89 SMN1; SMN2 (1.00) SMN1; SMN2GALR3CYP3A4CYP2C9NR2F2
SCHEMBL7264556 0.89 SMN1; SMN2 (0.78) SMN1; SMN2GALR3CYP3A4CYP2C9NR2F2
SCHEMBL7271947 0.89 SMN1; SMN2 (0.74) SMN1; SMN2GALR3CYP3A4CYP2C9NR2F2
Carboxyamidotriazole SCHEMBL8467240 0.88 SMN1; SMN2 (0.98) SMN1; SMN2GALR3CYP3A4CYP2C9NR2F2
SCHEMBL7264526 0.87 SMN1; SMN2 (0.80) SMN1; SMN2GALR3CYP3A4CYP2C9NR2F2
SCHEMBL7270852 0.86 SMN1; SMN2 (0.75) SMN1; SMN2GALR3CYP3A4CYP2C9NR2F2
SCHEMBL17507850 0.85 SMN1; SMN2 (0.88) SMN1; SMN2GALR3CYP3A4CYP2C9NR2F2
SCHEMBL7264241 0.84 SMN1; SMN2 (0.86) SMN1; SMN2GALR3CYP3A4CYP2C9NR2F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151529-B1 5-(AMINO OR SUBSTITUTED AMINO)-1,2,3-TRIAZOLES MERCK & CO. INC. (US) 1991-09-18 EP disclosed
US-4590201-A ANTICOCCIDIAL AGENT FOR ANIMALS PARTICULARLY FOR POULTRY MERCK & CO., INC. (US) 1986-05-20 US disclosed
EP-0151529-A2 5-(Amino or substituted amino)-1,2,3-triazoles MERCK & CO. INC. (US) 1985-08-14 EP disclosed