SCHEMBL7269053

SCHEMBL7269053

O=C(O)c1cnccc1Sc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 1/20 0.50
PTGS1 P23219 2/20 0.47
PTGS2 P35354 2/20 0.47
SLC22A12 Q96S37 4/20 0.46
KDM4C Q9H3R0 9/20 0.44
KDM4D Q6B0I6 4/20 0.44
KDM6B O15054 4/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 2/20 0.44
KDM4A O75164 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
THRB P10828 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HPGD P15428 1/20 0.44
NSD2 O96028 1/20 0.43
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5087701 0.87 SIRT1 (0.65) SIRT1PTGS1PTGS2SLC22A12KDM4E
SCHEMBL21056657 0.86 PTGS1 (0.50) SIRT1PTGS1PTGS2SLC22A12KDM4C
SCHEMBL30997714 0.86 PTGS1 (0.50) SIRT1PTGS1PTGS2SLC22A12KDM4C
Nitrous Acid SCHEMBL29269841 0.81 PTGS1 (0.46) SIRT1PTGS1PTGS2SLC22A12KDM4C
SCHEMBL1656950 0.80 POLB (0.52) SLC22A12KDM4CKDM4DKDM6BMEN1
SCHEMBL11504517 0.78 KDM4C (0.50) SLC22A12KDM4CKDM4DKDM6BMEN1
SCHEMBL231042 0.77 SIRT1 (0.71) SIRT1MEN1KMT2AKDM4EALDH1A1
SCHEMBL30997722 0.77 KDM4C (0.55) PTGS1PTGS2SLC22A12KDM4CKDM4D
SCHEMBL3074800 0.77 KDM4C (0.49) SLC22A12KDM4CKDM4DKDM6BMEN1
SCHEMBL10469069 0.76 CA12 (0.57) KDM4CKDM4DKDM6BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1360489-A1 LOW AFFINITY SCREENING METHOD Graffinity Pharmaceuticals Aktiengesellschaft (DE) 2003-11-12 EP disclosed
WO-2002063299-A1 LOW AFFINITY SCREENING METHOD GRAFFINITY PHARMACEUTICALS AG (DE) 2002-08-15 WO disclosed